[des-Arg10]kallidin

Ligand id: 644

Name: [des-Arg10]kallidin

Species: Human

Structure and Physico-chemical Properties

2D Structure
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Natural/Endogenous Targets
Target
B1 receptor
B2 receptor
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
B1 receptor Hs Agonist Full agonist 9.6 – 10.0 pKi - 1-3,6
pKi 9.6 – 10.0 [1-3,6]
B1 receptor Mm Agonist Full agonist 8.8 pKi - 5
pKi 8.8 [5]
B1 receptor Rn Agonist Full agonist 8.7 – 8.9 pKi - 6
pKi 8.7 – 8.9 [6]
B2 receptor Mm Agonist Partial agonist 4.6 pIC50 - 4
pIC50 4.6 [4]
Additional information and targets (data relate to human unless otherwise stated)
Description Data Reference
Ligand mentioned in the following text fields