AM-(20-50) (rat)   Click here for help

GtoPdb Ligand ID: 705

Synonyms: rat adrenomedullin (20-50)
Comment: Synthetic fragment of rat adrenomedullin
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
AM2 receptor Rn Antagonist Antagonist 7.8 pIC50 - 4
pIC50 7.8 [4]
AM1 receptor Rn Antagonist Antagonist 7.0 – 8.5 pIC50 - 1-2,4-5
pIC50 7.0 – 8.5 [1-2,4-5]
AM1 receptor Mm Antagonist Antagonist 7.5 pIC50 - 3
pIC50 7.5 [3]
AM2 receptor Mm Antagonist Antagonist 7.3 – 7.4 pIC50 - 3
pIC50 7.3 – 7.4 [3]