compound 1 [PMID: 25241924]   Click here for help

GtoPdb Ligand ID: 7801

Comment: Lipopeptide agonist of the apelin receptor. This palmitoylated peptide is the first of its kind found to be an agonist at this receptor.
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
apelin receptor Hs Agonist Full agonist 7.5 pEC50 - 1
pEC50 7.5 (EC50 3.37x10-8 M) [1]