compound 1 [PMID: 25241924]   Click here for help

GtoPdb Ligand ID: 7801

Comment: Lipopeptide agonist of the apelin receptor. This palmitoylated peptide is the first of its kind found to be an agonist at this receptor.
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1. McKeown SC, Zecri FJ, Fortier E, Taggart A, Sviridenko L, Adams CM, McAllister KH, Pin SS. (2014)
The design and implementation of a generic lipopeptide scanning platform to enable the identification of 'locally acting' agonists for the apelin receptor.
Bioorg Med Chem Lett, 24 (20): 4871-5. [PMID:25241924]