[125I]astressin   Click here for help

GtoPdb Ligand ID: 924

 Ligand is labelled  Ligand is radioactive
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
CRF1 receptor Hs Antagonist Antagonist 9.2 – 9.3 pKd - 1-2
pKd 9.2 – 9.3 [1-2]
CRF2 receptor Hs Antagonist Antagonist 9.6 – 9.7 pKi - 1-2
pKi 9.6 – 9.7 [1-2]