NNC1702   Click here for help

GtoPdb Ligand ID: 9760

Synonyms: des-His1-[Glu9, Lys24(4 X γGlu), Leu27]glucagon
Comment: Low-potency partial agonist, designed to have reduced agonist activity but to maintain relatively high binding affinity to the receptor [1].
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
glucagon receptor Hs Agonist Agonist 7.3 pIC50 - 1
pIC50 7.3 (IC50 5.35x10-8 M) [1]