Synonyms: Optimine® | SCH-10649
azatadine is an approved drug (FDA (1977))
Compound class:
Synthetic organic
Comment: Azatadine is a first-generation antihistamine and anticholinergic drug. Its marketing has been discontinued in many countries as its use has largely been repleaced by newer and more effective alternatives.
![]() Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
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No information available. |
Summary of Clinical Use ![]() |
Used to reduce symptoms of allergies (such as sneezing, itching, runny nose and watery eyes, rashes). |
Mechanism Of Action and Pharmacodynamic Effects ![]() |
Azatadine blocks the action of endogenous histamine at the histamine H1 receptor. |