Synonyms: BTT 3033 | BTT3033
Compound class:
Synthetic organic
Comment: BTT-3033 is an α2β1 integrin inhibitor that blocks platelet attachment to collagen [1].
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References |
1. Nissinen L, Koivunen J, Käpylä J, Salmela M, Nieminen J, Jokinen J, Sipilä K, Pihlavisto M, Pentikäinen OT, Marjamäki A et al.. (2012)
Novel α2β1 integrin inhibitors reveal that integrin binding to collagen under shear stress conditions does not require receptor preactivation. J Biol Chem, 287 (53): 44694-702. [PMID:23132859] |