[Phe(Me)7]neurokinin B   Click here for help

GtoPdb Ligand ID: 2113

Synonyms: [MePhe7]NKB
Comment: Synthetic analogue of neurokinin B
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1. Chung FZ, Wu LH, Tian Y, Vartanian MA, Lee H, Bikker J, Humblet C, Pritchard MC, Raphy J, Suman-Chauhan N. (1995)
Two classes of structurally different antagonists display similar species preference for the human tachykinin neurokinin3 receptor.
Mol Pharmacol, 48 (4): 711-6. [PMID:7476898]
2. Drapeau G, Rouissi N, Nantel F, Rhaleb NE, Tousignant C, Regoli D. (1990)
Antagonists for the neurokinin NK-3 receptor evaluated in selective receptor systems.
Regul Pept, 31 (2): 125-35. [PMID:2176308]
3. Sarau HM, Feild JA, Ames RS, Foley JJ, Nuthulaganti P, Schmidt DB, Buckley PT, Elshourbagy NA, Brawner ME, Luttmann MA et al.. (2001)
Molecular and pharmacological characterization of the murine tachykinin NK(3) receptor.
Eur J Pharmacol, 413 (2-3): 143-50. [PMID:11226387]
4. Sarau HM, Griswold DE, Potts W, Foley JJ, Schmidt DB, Webb EF, Martin LD, Brawner ME, Elshourbagy NA, Medhurst AD et al.. (1997)
Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.
J Pharmacol Exp Ther, 281 (3): 1303-11. [PMID:9190866]