tertiapin-Q   

GtoPdb Ligand ID: 2383

Synonyms: TPN(Q)
Comment: From the venom gland of Apis mellifera (honeybee)
References
1. Felix JP, Liu J, Schmalhofer WA, Bailey T, Bednarek MA, Kinkel S, Weinglass AB, Kohler M, Kaczorowski GJ, Priest BT, Garcia ML. (2006)
Characterization of Kir1.1 channels with the use of a radiolabeled derivative of tertiapin.
Biochemistry, 45 (33): 10129-39. [PMID:16906771]
2. Jin W, Klem AM, Lewis JH, Lu Z. (1999)
Mechanisms of inward-rectifier K+ channel inhibition by tertiapin-Q.
Biochemistry, 38 (43): 14294-301. [PMID:10572004]
3. Jin W, Lu Z. (1998)
A novel high-affinity inhibitor for inward-rectifier K+ channels.
Biochemistry, 37 (38): 13291-9. [PMID:9748337]
4. Jin W, Lu Z. (1999)
Synthesis of a stable form of tertiapin: a high-affinity inhibitor for inward-rectifier K+ channels.
Biochemistry, 38 (43): 14286-93. [PMID:10572003]