Synonyms: galanin(1-13)spantide
Compound class:
Peptide
![]() Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
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References |
1. Bloomquist BT, Beauchamp MR, Zhelnin L, Brown SE, Gore-Willse AR, Gregor P, Cornfield LJ. (1998)
Cloning and expression of the human galanin receptor GalR2. Biochem Biophys Res Commun, 243 (2): 474-9. [PMID:9480833] |
2. Borowsky B, Walker MW, Huang LY, Jones KA, Smith KE, Bard J, Branchek TA, Gerald C. (1998)
Cloning and characterization of the human galanin GALR2 receptor. Peptides, 19 (10): 1771-81. [PMID:9880084] |
3. Fathi Z, Battaglino PM, Iben LG, Li H, Baker E, Zhang D, McGovern R, Mahle CD, Sutherland GR, Iismaa TP et al.. (1998)
Molecular characterization, pharmacological properties and chromosomal localization of the human GALR2 galanin receptor. Brain Res Mol Brain Res, 58 (1-2): 156-69. [PMID:9685625] |
4. Fathi Z, Cunningham AM, Iben LG, Battaglino PB, Ward SA, Nichol KA, Pine KA, Wang J, Goldstein ME, Iismaa TP et al.. (1997)
Cloning, pharmacological characterization and distribution of a novel galanin receptor. Brain Res Mol Brain Res, 51 (1-2): 49-59. [PMID:9427506] |
5. Fitzgerald LW, Patterson JP, Conklin DS, Horlick R, Largent BL. (1998)
Pharmacological and biochemical characterization of a recombinant human galanin GALR1 receptor: agonist character of chimeric galanin peptides. J Pharmacol Exp Ther, 287 (2): 448-56. [PMID:9808667] |
6. Howard AD, Tan C, Shiao LL, Palyha OC, McKee KK, Weinberg DH, Feighner SD, Cascieri MA, Smith RG, Van Der Ploeg LH et al.. (1997)
Molecular cloning and characterization of a new receptor for galanin. FEBS Lett, 405 (3): 285-90. [PMID:9108306] |
7. Pang L, Hashemi T, Lee HJ, Maguire M, Graziano MP, Bayne M, Hawes B, Wong G, Wang S. (1998)
The mouse GalR2 galanin receptor: genomic organization, cDNA cloning, and functional characterization. J Neurochem, 71 (6): 2252-9. [PMID:9832122] |
8. Parker EM, Izzarelli DG, Nowak HP, Mahle CD, Iben LG, Wang J, Goldstein ME. (1995)
Cloning and characterization of the rat GALR1 galanin receptor from Rin14B insulinoma cells. Brain Res Mol Brain Res, 34 (2): 179-89. [PMID:8750821] |
9. Smith KE, Forray C, Walker MW, Jones KA, Tamm JA, Bard J, Branchek TA, Linemeyer DL, Gerald C. (1997)
Expression cloning of a rat hypothalamic galanin receptor coupled to phosphoinositide turnover. J Biol Chem, 272 (39): 24612-6. [PMID:9305929] |
10. Smith KE, Walker MW, Artymyshyn R, Bard J, Borowsky B, Tamm JA, Yao WJ, Vaysse PJ, Branchek TA, Gerald C et al.. (1998)
Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem, 273 (36): 23321-6. [PMID:9722565] |
11. Sullivan KA, Shiao LL, Cascieri MA. (1997)
Pharmacological characterization and tissue distribution of the human and rat GALR1 receptors. Biochem Biophys Res Commun, 233 (3): 823-8. [PMID:9168941] |
12. Wang S, Hashemi T, He C, Strader C, Bayne M. (1997)
Molecular cloning and pharmacological characterization of a new galanin receptor subtype. Mol Pharmacol, 52 (3): 337-43. [PMID:9281594] |
13. Wang S, He C, Hashemi T, Bayne M. (1997)
Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes. J Biol Chem, 272 (51): 31949-52. [PMID:9405385] |
14. Wang S, He C, Maguire MT, Clemmons AL, Burrier RE, Guzzi MF, Strader CD, Parker EM, Bayne ML. (1997)
Genomic organization and functional characterization of the mouse GalR1 galanin receptor. FEBS Lett, 411 (2-3): 225-30. [PMID:9271210] |