R3(BΔ23-27)R/I5 chimeric peptide

Ligand id: 3907

Name: R3(BΔ23-27)R/I5 chimeric peptide

References
1. Haugaard-Kedström LM, Shabanpoor F, Hossain MA, Clark RJ, Ryan PJ, Craik DJ, Gundlach AL, Wade JD, Bathgate RA, Rosengren KJ. (2011)
Design, synthesis, and characterization of a single-chain peptide antagonist for the relaxin-3 receptor RXFP3.
J. Am. Chem. Soc., 133 (13): 4965-74. [PMID:21384867]
2. Kocan M, Sarwar M, Hossain MA, Wade JD, Summers RJ. (2014)
Signalling profiles of H3 relaxin, H2 relaxin and R3(BΔ23-27)R/I5 acting at the relaxin family peptide receptor 3 (RXFP3).
Br. J. Pharmacol., 171 (11): 2827-41. [PMID:24641548]
3. Kuei C, Sutton S, Bonaventure P, Pudiak C, Shelton J, Zhu J, Nepomuceno D, Wu J, Chen J, Kamme F et al.. (2007)
R3(BDelta23 27)R/I5 chimeric peptide, a selective antagonist for GPCR135 and GPCR142 over relaxin receptor LGR7: in vitro and in vivo characterization.
J. Biol. Chem., 282 (35): 25425-35. [PMID:17606621]