Synonyms: [3H]-CGS21680
Compound class:
Synthetic organic
Comment: The position of the tritiated hydrogen(s) is not specified in the available literature therefore our structure does not show the position of the radiolabel.
![]() Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
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References |
1. Jarvis MF, Schulz R, Hutchison AJ, Do UH, Sills MA, Williams M. (1989)
[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain. J Pharmacol Exp Ther, 251 (3): 888-93. [PMID:2600819] |
2. Wan W, Sutherland GR, Geiger JD. (1990)
Binding of the adenosine A2 receptor ligand [3H]CGS 21680 to human and rat brain: evidence for multiple affinity sites. J Neurochem, 55 (5): 1763-71. [PMID:2213023] |