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Compound class: Peptide or derivative
Ligand Activity Visualisation Charts
These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.✖
1. Bloomquist BT, Beauchamp MR, Zhelnin L, Brown SE, Gore-Willse AR, Gregor P, Cornfield LJ. (1998)
Cloning and expression of the human galanin receptor GalR2.
Biochem. Biophys. Res. Commun., 243 (2): 474-9. [PMID:9480833]
2. Howard AD, Tan C, Shiao LL, Palyha OC, McKee KK, Weinberg DH, Feighner SD, Cascieri MA, Smith RG, Van Der Ploeg LH et al.. (1997)
Molecular cloning and characterization of a new receptor for galanin.
FEBS Lett., 405 (3): 285-90. [PMID:9108306]
3. Pang L, Hashemi T, Lee HJ, Maguire M, Graziano MP, Bayne M, Hawes B, Wong G, Wang S. (1998)
The mouse GalR2 galanin receptor: genomic organization, cDNA cloning, and functional characterization.
J. Neurochem., 71 (6): 2252-9. [PMID:9832122]
4. Sullivan KA, Shiao LL, Cascieri MA. (1997)
Pharmacological characterization and tissue distribution of the human and rat GALR1 receptors.
Biochem. Biophys. Res. Commun., 233 (3): 823-8. [PMID:9168941]
5. Wang S, Ghibaudi L, Hashemi T, He C, Strader C, Bayne M, Davis H, Hwa JJ. (1998)
The GalR2 galanin receptor mediates galanin-induced jejunal contraction, but not feeding behavior, in the rat: differentiation of central and peripheral effects of receptor subtype activation.
FEBS Lett., 434 (3): 277-82. [PMID:9742938]
6. Wang S, He C, Hashemi T, Bayne M. (1997)
Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes.
J. Biol. Chem., 272 (51): 31949-52. [PMID:9405385]