GAL2 receptor
|
|
|
Hs |
Agonist |
Agonist |
<6.2 |
pKi |
- |
1 |
|
⤷ |
pKi
<6.2
(Ki >7x10-7 M)
[1]
|
GAL1 receptor
|
|
|
Rn |
Agonist |
Agonist |
<6.0 |
pKi |
- |
5-6 |
|
⤷ |
pKi
<6.0
(Ki >1x10-6 M)
[5-6]
|
GAL3 receptor
|
|
|
Rn |
Agonist |
Agonist |
<6.0 |
pKi |
- |
5-6 |
|
⤷ |
pKi
<6.0
(Ki >1x10-6 M)
[5-6]
|
GAL1 receptor
|
|
|
Mm |
Agonist |
Agonist |
<5.8 |
pKi |
- |
3 |
|
⤷ |
pKi
<5.8
(Ki >1.65x10-6 M)
[3]
|
GAL2 receptor
|
|
|
Rn |
Agonist |
Agonist |
5.5 – 6.0 |
pKi |
- |
3,5-6 |
|
⤷ |
pKi
5.5 – 6.0
(Ki 3.125x10-6 – 1x10-6 M)
[3,5-6]
|
GAL2 receptor
|
|
|
Mm |
Agonist |
Agonist |
<5.7 |
pKi |
- |
3 |
|
⤷ |
pKi
<5.7
(Ki >2.2x10-6 M)
[3]
|
GAL1 receptor
|
|
|
Hs |
Agonist |
Agonist |
<6.0 |
pIC50 |
- |
4 |
|
⤷ |
pIC50
<6.0
(IC50 >1x10-6 M)
[4]
|
GAL1 receptor
|
|
|
Rn |
Agonist |
Agonist |
<6.0 |
pIC50 |
- |
2,4 |
|
⤷ |
pIC50
<6.0
(IC50 >1x10-6 M)
[2,4]
|
GAL2 receptor
|
|
|
Rn |
Agonist |
Agonist |
<6.0 |
pIC50 |
- |
2 |
|
⤷ |
pIC50
<6.0
(IC50 >1x10-6 M)
[2]
|