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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fms related receptor tyrosine kinase 3 in Human [GtoPdb: 1807] [UniProtKB: P36888] | ||||||||
| GtoPdb | - | - | 7.21 | pIC50 | 62 | nM | IC50 | J Med Chem (2020) 63: 14921-14936 [PMID:33256400] |
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | - | - | 7.38 | pIC50 | 42 | nM | IC50 | J Med Chem (2020) 63: 14921-14936 [PMID:33256400] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | Inhibitory effect in a biochemical enzyme assay | - | 8.52 | pIC50 | 3 | nM | IC50 | J Med Chem (2020) 63: 14921-14936 [PMID:33256400] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 7.03 | pIC50 | 94 | nM | IC50 | J Med Chem (2020) 63: 14921-14936 [PMID:33256400] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | - | - | 7.12 | pIC50 | 75 | nM | IC50 | J Med Chem (2020) 63: 14921-14936 [PMID:33256400] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.