m-chlorophenylpiperazine [Ligand Id: 142] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL478 (1-M-Chlorophenyl Piperazine Metabolite, Chlorophenylpiperazine, mCPP) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| β1-adrenoceptor/Beta-1 adrenergic receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL213] [GtoPdb: 28] [UniProtKB: P08588] | ||||||||
| ChEMBL | Binding affinity for Beta-1 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine ventricular muscle in the presence of 1 uM zinterol | B | 5.7 | pIC50 | 2000 | nM | IC50 | J Med Chem (1992) 35: 743-750 [PMID:1347318] |
| Beta-2 adrenergic receptor in Dog (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2289] [UniProtKB: P54833] | ||||||||
| ChEMBL | Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung tissue in the presence of 0.1 uM metoprolol | B | 4.74 | pIC50 | 18000 | nM | IC50 | J Med Chem (1992) 35: 743-750 [PMID:1347318] |
| D1 receptor/Dopamine D1 receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL265] [GtoPdb: 214] [UniProtKB: P18901] | ||||||||
| ChEMBL | Binding affinity at rat Dopamine receptor D1 by [3H]SCH-23390 displacement. | B | 6 | pKi | >1000 | nM | Ki | J Med Chem (1989) 32: 1052-1056 [PMID:2565400] |
| D2 receptor/Dopamine D2 receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL339] [GtoPdb: 215] [UniProtKB: P61169] | ||||||||
| ChEMBL | Binding affinity against rat Dopamine receptor D2. | B | 6 | pKi | >1000 | nM | Ki | J Med Chem (1989) 32: 1052-1056 [PMID:2565400] |
| 5-HT1A receptor/Serotonin 1a (5-HT1a) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL214] [GtoPdb: 1] [UniProtKB: P08908] | ||||||||
| ChEMBL | Binding affinity to 5HT1A receptor | B | 7 | pKd | 100 | nM | Kd | J Med Chem (2009) 52: 6107-6125 [PMID:19754201] |
| 5-HT1A receptor/Serotonin 1a (5-HT1a) receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL273] [GtoPdb: 1] [UniProtKB: P19327] | ||||||||
| ChEMBL | Evaluated for the binding affinity to hippocampus striatal membranes at 5-hydroxytryptamine 1A receptor binding site by using [3H]-8-OH- DPAT as a radioligand. | B | 5.62 | pKi | 2400 | nM | Ki | J Med Chem (1987) 30: 1-12 [PMID:3543362] |
| ChEMBL | Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenate (experiment 1) | B | 6.7 | pKi | 200 | nM | Ki | J Med Chem (1993) 36: 2751-2760 [PMID:8410989] |
| ChEMBL | Binding affinity of a compound to rat brain 5-hydroxytryptamine 1A (serotonin) receptor assayed by radiolabeled [3H]-8-OH-DPAT ligand displacement | B | 6.84 | pKi | 144.54 | nM | Ki | J Med Chem (1996) 39: 126-134 [PMID:8568799] |
| ChEMBL | Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenate (experiment 2) | B | 6.84 | pKi | 143 | nM | Ki | J Med Chem (1993) 36: 2751-2760 [PMID:8410989] |
| ChEMBL | In vitro ability to displace [3H]8-hydroxy-2-(di-n-propylamino) tetralin binding from 5-hydroxytryptamine 1A receptor site in rat brain hippocampus | B | 6.84 | pKi | 143 | nM | Ki | J Med Chem (1992) 35: 2369-2374 [PMID:1535661] |
| ChEMBL | Binding affinity towards rat 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT radioligand. | B | 6.89 | pKi | 130 | nM | Ki | J Med Chem (1996) 39: 4439-4450 [PMID:8893838] |
| ChEMBL | Evaluated for binding affinity towards 5-hydroxytryptamine 1A receptor in rat brain | B | 6.89 | pKi | 130 | nM | Ki | J Med Chem (1988) 31: 1968-1971 [PMID:3172131] |
| ChEMBL | Binding affinity at rat 5-hydroxytryptamine 1A receptor by [3H]WB-4101 displacement. | B | 7.64 | pKi | 23 | nM | Ki | J Med Chem (1989) 32: 1052-1056 [PMID:2565400] |
| 5-HT1B receptor/Serotonin 1b (5-HT1b) receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3459] [GtoPdb: 2] [UniProtKB: P28564] | ||||||||
| ChEMBL | Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand. | B | 7.12 | pKi | 75 | nM | Ki | J Med Chem (1987) 30: 1-12 [PMID:3543362] |
| ChEMBL | Binding affinity at rat 5-hydroxytryptamine 1B receptor by [3H]5-HT displacement. | B | 8.36 | pKi | 4.4 | nM | Ki | J Med Chem (1989) 32: 1052-1056 [PMID:2565400] |
| 5-HT2A receptor/Serotonin 2a (5-HT2a) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL224] [GtoPdb: 6] [UniProtKB: P28223] | ||||||||
| ChEMBL | Binding affinity to 5HT2A (unknown origin) | B | 6.56 | pKi | 273 | nM | Ki | Bioorg Med Chem Lett (2016) 26: 914-920 [PMID:26748694] |
| ChEMBL | Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell line | B | 7.27 | pKi | 54 | nM | Ki | Bioorg Med Chem Lett (2004) 14: 2367-2370 [PMID:15081042] |
| ChEMBL | Displacement of [125I]DOI from human 5HT2A | B | 7.27 | pKi | 54 | nM | Ki | Bioorg Med Chem Lett (2006) 16: 677-680 [PMID:16257207] |
| ChEMBL | Displacement of [125I]DOI from human recombinant 5HT2A expressed in HEK293E cells | B | 7.32 | pKi | 48 | nM | Ki | J Med Chem (2007) 50: 1365-1379 [PMID:17315987] |
| ChEMBL | Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293E cells | B | 7.32 | pKi | 48 | nM | Ki | Bioorg Med Chem Lett (2010) 20: 1128-1133 [PMID:20022752] |
| GtoPdb | - | - | 7.5 | pKi | - | - | - |
Naunyn Schmiedebergs Arch Pharmacol (2004) 370: 114-23 [PMID:15322733]; Biochem Pharmacol (1996) 51: 71-6 [PMID:8534270]; Naunyn Schmiedebergs Arch Pharmacol (1999) 359: 1-6 [PMID:9933142] |
| ChEMBL | Agonist activity at human recombinant 5HT2A receptor expressed in HEK293E cells by FLIPR assay | F | 6.54 | pEC50 | 290 | nM | EC50 | Bioorg Med Chem Lett (2010) 20: 1128-1133 [PMID:20022752] |
| ChEMBL | Activity at human 5HT2A expressed in HEK293E cells assessed as elevation of intracellular calcium by 384-FLIPR assay | F | 6.54 | pEC50 | 290 | nM | EC50 | J Med Chem (2007) 50: 1365-1379 [PMID:17315987] |
| ChEMBL | Agonist activity at human recombinant 5HT2A receptor expressed in Swiss mouse 3T3 cells assessed as induction of calcium mobilization by FLIPR assay | F | 6.78 | pEC50 | 167 | nM | EC50 | Bioorg Med Chem Lett (2009) 19: 5791-5795 [PMID:19716297] |
| ChEMBL | Binding to human 5HT2A receptor expressed in CHO cells | B | 7.12 | pEC50 | 75 | nM | EC50 | Bioorg Med Chem Lett (2006) 16: 677-680 [PMID:16257207] |
| ChEMBL | Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate reader | F | 7.12 | pEC50 | 75 | nM | EC50 | Bioorg Med Chem Lett (2004) 14: 2367-2370 [PMID:15081042] |
| ChEMBL | Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as intracellular IP3 accumulation | F | 7.2 | pEC50 | 63.1 | nM | EC50 | J Med Chem (2008) 51: 305-313 [PMID:18095642] |
| ChEMBL | Agonist activity at serotonin-activated human recombinant 5HT-2A receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins measured for 1 min by fluorescence assay | F | 8.14 | pEC50 | 7.2 | nM | EC50 | Eur J Med Chem (2013) 63: 558-569 [PMID:23537943] |
| 5-HT2A receptor in Rat [GtoPdb: 6] [UniProtKB: P14842] | ||||||||
| GtoPdb | - | - | 6.4 | pKi | - | - | - | Circulation (2000) 102: 2836-41 [PMID:11104741] |
| 5-HT2B receptor/Serotonin 2b (5-HT2b) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1833] [GtoPdb: 7] [UniProtKB: P41595] | ||||||||
| ChEMBL | Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell line | B | 7.49 | pKi | 32 | nM | Ki | Bioorg Med Chem Lett (2004) 14: 2367-2370 [PMID:15081042] |
| ChEMBL | Displacement of [3H]5-HT from human 5HT2B | B | 7.49 | pKi | 32 | nM | Ki | Bioorg Med Chem Lett (2006) 16: 677-680 [PMID:16257207] |
| ChEMBL | Displacement of [3H]LSD from human recombinant 5HT2B expressed in HEK293E cells | B | 7.62 | pKi | 24 | nM | Ki | J Med Chem (2007) 50: 1365-1379 [PMID:17315987] |
| ChEMBL | Displacement of [125I]LSD from human recombinant 5HT2B receptor expressed in HEK293E cells | B | 7.62 | pKi | 24 | nM | Ki | Bioorg Med Chem Lett (2010) 20: 1128-1133 [PMID:20022752] |
| GtoPdb | - | - | 8.5 | pKi | - | - | - |
Naunyn Schmiedebergs Arch Pharmacol (2004) 370: 114-23 [PMID:15322733]; Circulation (2000) 102: 2836-41 [PMID:11104741]; Naunyn Schmiedebergs Arch Pharmacol (1999) 359: 1-6 [PMID:9933142]; Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 17-24 [PMID:9459568]; Br J Pharmacol (2003) 140: 277-84 [PMID:12970106] |
| ChEMBL | Binding to human 5HT2B receptor expressed in CHO cells | B | 6 | pEC50 | >1000 | nM | EC50 | Bioorg Med Chem Lett (2006) 16: 677-680 [PMID:16257207] |
| ChEMBL | Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate reader | F | 6 | pEC50 | >1000 | nM | EC50 | Bioorg Med Chem Lett (2004) 14: 2367-2370 [PMID:15081042] |
| ChEMBL | Agonist activity at human recombinant 5HT2B receptor expressed in HEK293E cells by FLIPR assay | F | 6.54 | pEC50 | 287 | nM | EC50 | Bioorg Med Chem Lett (2010) 20: 1128-1133 [PMID:20022752] |
| ChEMBL | Activity at human 5HT2B expressed in HEK293E cells assessed as elevation of intracellular calcium by 384-FLIPR assay | F | 6.54 | pEC50 | 287 | nM | EC50 | J Med Chem (2007) 50: 1365-1379 [PMID:17315987] |
| ChEMBL | Agonist activity at human recombinant 5HT2B receptor expressed in Swiss mouse 3T3 cells assessed as induction of calcium mobilization by FLIPR assay | F | 6.9 | pEC50 | 125 | nM | EC50 | Bioorg Med Chem Lett (2009) 19: 5791-5795 [PMID:19716297] |
| ChEMBL | Agonist activity at human recombinant 5HT2B receptor assessed as induction of calcium mobilization by FLIPR assay | F | 6.9 | pEC50 | 125 | nM | EC50 | Bioorg Med Chem Lett (2009) 19: 4999-5003 [PMID:19646865] |
| ChEMBL | Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as intracellular IP3 accumulation | F | 7.4 | pEC50 | 39.81 | nM | EC50 | J Med Chem (2008) 51: 305-313 [PMID:18095642] |
| 5-HT2B receptor in Rat [GtoPdb: 7] [UniProtKB: P30994] | ||||||||
| GtoPdb | - | - | 7.6 | pKi | - | - | - | Mol Pharmacol (1993) 43: 419-26 [PMID:8450835] |
| 5-HT2C receptor/Serotonin 2c (5-HT2c) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL225] [GtoPdb: 8] [UniProtKB: P28335] | ||||||||
| ChEMBL | Binding affinity to 5HT2C (unknown origin) | B | 7.56 | pKi | 27.7 | nM | Ki | Bioorg Med Chem Lett (2016) 26: 914-920 [PMID:26748694] |
| ChEMBL | Displacement of [125I]DOI from human recombinant 5HT2C expressed in HEK293E cells | B | 7.77 | pKi | 17 | nM | Ki | J Med Chem (2007) 50: 1365-1379 [PMID:17315987] |
| ChEMBL | Displacement of [125I]DOI from human recombinant 5HT2C receptor expressed in HEK293E cells | B | 7.77 | pKi | 17 | nM | Ki | Bioorg Med Chem Lett (2010) 20: 1128-1133 [PMID:20022752] |
| ChEMBL | Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell line | B | 8.05 | pKi | 9 | nM | Ki | Bioorg Med Chem Lett (2004) 14: 2367-2370 [PMID:15081042] |
| ChEMBL | Displacement of [3H]5-HT from human 5HT2C | B | 8.05 | pKi | 9 | nM | Ki | Bioorg Med Chem Lett (2006) 16: 677-680 [PMID:16257207] |
| ChEMBL | Displacement of [125I]DOI from recombinant human 5-HT2C receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting | B | 8.1 | pKi | 7.94 | nM | Ki | Bioorg Med Chem Lett (2016) 26: 5877-5882 [PMID:27864071] |
| GtoPdb | - | - | 8.5 | pKi | - | - | - |
Naunyn Schmiedebergs Arch Pharmacol (2004) 370: 114-23 [PMID:15322733]; Naunyn Schmiedebergs Arch Pharmacol (1999) 359: 1-6 [PMID:9933142]; Br J Pharmacol (2003) 140: 277-84 [PMID:12970106]; J Neurochem (1999) 72: 2127-34 [PMID:10217294]; Synapse (2000) 35: 144-150 [PMID:10611640]; Eur J Pharmacol (2004) 483: 37-43 [PMID:14709324] |
| ChEMBL | Agonist activity at human recombinant 5HT2C receptor expressed in CHO K1 cells assessed as induction of calcium mobilization by FLIPR assay | F | 6.77 | pEC50 | 170 | nM | EC50 | Bioorg Med Chem Lett (2009) 19: 4999-5003 [PMID:19646865] |
| ChEMBL | Agonist activity at human recombinant 5HT2C receptor expressed in CHOK1 cells assessed as induction of calcium mobilization by FLIPR assay | F | 6.77 | pEC50 | 170 | nM | EC50 | Bioorg Med Chem Lett (2009) 19: 5791-5795 [PMID:19716297] |
| ChEMBL | Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometric imaging plate reader | F | 7.59 | pEC50 | 26 | nM | EC50 | Bioorg Med Chem Lett (2004) 14: 2367-2370 [PMID:15081042] |
| ChEMBL | Binding to human 5HT2C receptor expressed in CHO cells | B | 7.59 | pEC50 | 26 | nM | EC50 | Bioorg Med Chem Lett (2006) 16: 677-680 [PMID:16257207] |
| ChEMBL | Activity at human 5HT2C expressed in HEK293E cells assessed as elevation of intracellular calcium by 384-FLIPR assay | F | 7.82 | pEC50 | 15 | nM | EC50 | J Med Chem (2007) 50: 1365-1379 [PMID:17315987] |
| ChEMBL | Agonist activity at human recombinant 5HT2C receptor expressed in HEK293E cells by FLIPR assay | F | 7.82 | pEC50 | 15 | nM | EC50 | Bioorg Med Chem Lett (2010) 20: 1128-1133 [PMID:20022752] |
| ChEMBL | Agonist activity at recombinant human 5-HT2C receptor expressed in HEK293E cells assessed as induction of intracellular Ca2+ levels after 90 secs by Fluo-4-dye based FLIPR assay | F | 7.82 | pEC50 | 15 | nM | EC50 | J Med Chem (2017) 60: 6166-6190 [PMID:28635286] |
| ChEMBL | Agonist activity at unedited 5-HT2C receptor (unknown origin) expressed in HEK293 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by scintillation counting | F | 7.9 | pEC50 | 12.59 | nM | EC50 | Bioorg Med Chem Lett (2016) 26: 5877-5882 [PMID:27864071] |
| ChEMBL | Agonist activity at serotonin-activated human recombinant 5HT-2C receptor expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins measured for 1 min by fluorescence assay | F | 8.09 | pEC50 | 8.1 | nM | EC50 | Eur J Med Chem (2013) 63: 558-569 [PMID:23537943] |
| ChEMBL | Agonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as intracellular IP3 accumulation | F | 8.1 | pEC50 | 7.94 | nM | EC50 | J Med Chem (2008) 51: 305-313 [PMID:18095642] |
| 5-HT2C receptor in Rat [GtoPdb: 8] [UniProtKB: P08909] | ||||||||
| GtoPdb | - | - | 7.2 | pKi | - | - | - | Circulation (2000) 102: 2836-41 [PMID:11104741] |
| 5-HT3E/5-HT3B/5-HT3A/5-HT3D/5-HT3C/Serotonin 3 (5-HT3) receptor in Human (target type: PROTEIN COMPLEX GROUP) [ChEMBL: CHEMBL2094132] [GtoPdb: 377, 374, 373, 376, 375] [UniProtKB: A5X5Y0, O95264, P46098, Q70Z44, Q8WXA8] | ||||||||
| ChEMBL | Compound was tested for the inhibition of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor expressed in NG 108-15 cells | B | 7.21 | pKi | 62 | nM | Ki | J Med Chem (1996) 39: 4017-4026 [PMID:8831767] |
| 5-HT5A receptor/Serotonin 5a (5-HT5a) receptor in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3597] [GtoPdb: 10] [UniProtKB: P30966] | ||||||||
| ChEMBL | Binding affinity towards murine 5-hydroxytryptamine 5A receptor | B | 5.06 | pKi | 8700 | nM | Ki | J Med Chem (2003) 46: 2795-2812 [PMID:12825922] |
| ChEMBL | Binding affinity towards mouse 5-hydroxytryptamine 5A receptor was evaluated using [3H]LSD as radioligand | B | 5.06 | pKi | 8700 | nM | Ki | J Med Chem (2003) 46: 2795-2812 [PMID:12825922] |
| 5-HT6 receptor/Serotonin 6 (5-HT6) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3371] [GtoPdb: 11] [UniProtKB: P50406] | ||||||||
| ChEMBL | Binding affinity towards human 5-hydroxytryptamine 6 receptor was evaluated using [125I]-2-iodo LSD as radioligand | B | 5.64 | pKi | 2300 | nM | Ki | J Med Chem (2003) 46: 2795-2812 [PMID:12825922] |
| 5-HT6 receptor in Rat [GtoPdb: 11] [UniProtKB: P31388] | ||||||||
| GtoPdb | - | - | 5.6 | pKi | - | - | - | Mol Pharmacol (1993) 43: 320-7 [PMID:7680751] |
| 5-HT7 receptor/Serotonin 7 (5-HT7) receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3155] [GtoPdb: 12] [UniProtKB: P34969] | ||||||||
| ChEMBL | Binding affinity of compound towards rodent 5-hydroxytryptamine 7 receptor | B | 6.52 | pKi | 304 | nM | Ki | J Med Chem (2003) 46: 2795-2812 [PMID:12825922] |
| 5-HT7 receptor/Serotonin 7 (5-HT7) receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3223] [GtoPdb: 12] [UniProtKB: P32305] | ||||||||
| ChEMBL | Displacement of [3H]LSD from rat kidney proximal convoluted tubule 5HT7R expressed in COS7 cells | B | 6.45 | pKi | 352 | nM | Ki | J Med Chem (2012) 55: 6375-6380 [PMID:22738316] |
| GtoPdb | - | - | 6.6 | pKi | - | - | - | J Biol Chem (1993) 268: 18200-4 [PMID:8394362] |
| SERT/Serotonin transporter in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL228] [GtoPdb: 928] [UniProtKB: P31645] | ||||||||
| ChEMBL | Binding affinity to SERT (unknown origin) | B | 6.57 | pKi | 271 | nM | Ki | Bioorg Med Chem Lett (2016) 26: 914-920 [PMID:26748694] |
| sigma non-opioid intracellular receptor 1/Sigma opioid receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL287] [GtoPdb: 2552] [UniProtKB: Q99720] | ||||||||
| ChEMBL | Binding affinity towards sigma receptor in guinea pig brain membranes using [3H]DTG as radioligand | B | 5.21 | pKi | 6150 | nM | Ki | J Med Chem (1991) 34: 3360-3365 [PMID:1662725] |
| 5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221] | ||||||||
| GtoPdb | - | - | 6.7 | pKi | - | - | - | Mol Pharmacol (1991) 40: 143-8 [PMID:1652050] |
| 5-ht1e receptor in Human [GtoPdb: 4] [UniProtKB: P28566] | ||||||||
| GtoPdb | - | - | 5.4 | pKi | - | - | - | Eur J Pharmacol (2004) 484: 127-39 [PMID:14744596] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
