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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
LPA4 receptor in Human [GtoPdb: 94] [UniProtKB: Q99677] | ||||||||
GtoPdb | - | - | 5.7 | pIC50 | - | - | - | J Biol Chem (2009) 284: 17304-19 [PMID:19366702] |
LPA5 receptor in Human [GtoPdb: 124] [UniProtKB: Q9H1C0] | ||||||||
GtoPdb | - | - | 6.54 | pEC50 | 290 | nM | EC50 |
J Biol Chem (2009) 284: 17304-19 [PMID:19366702]; J Biol Chem (2008) 283: 21054-64 [PMID:18499677] |
LPA2 receptor in Human [GtoPdb: 273] [UniProtKB: Q9HBW0] | ||||||||
GtoPdb | - | - | 5.68 | pIC50 | - | - | - | J Biol Chem (2009) 284: 17304-19 [PMID:19366702] |
LPA3 receptor in Human [GtoPdb: 274] [UniProtKB: Q9UBY5] | ||||||||
GtoPdb | - | - | 6.81 | pKd | - | - | - | Biochim Biophys Acta (2006) 1761: 1506-14 [PMID:17092771] |
GtoPdb | - | - | 6.81 | pIC50 | - | - | - | J Biol Chem (2009) 284: 17304-19 [PMID:19366702] |
TRPV3 in Mouse [GtoPdb: 509] [UniProtKB: Q8K424] | ||||||||
GtoPdb | Calcium imaging and patch clamp electrophysiology | - | 6.89 | pEC50 | 130 | nM | EC50 | J Biol Chem (2010) 285: 19362-71 [PMID:20395302] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.