Mg2+ [Ligand Id: 708] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CaS receptor in Rat [GtoPdb: 54] [UniProtKB: P48442] | ||||||||
| GtoPdb | - | - | 2.4 | pKd | - | - | - |
Proc Natl Acad Sci USA (1995) 92: 131-5 [PMID:7816802]; Bone Miner (1989) 5: 249-57 [PMID:2655774] |
| HCN1 in Mouse [GtoPdb: 400] [UniProtKB: O88704] | ||||||||
| GtoPdb | - | - | 3.3 | pIC50 | - | - | - | Am J Physiol, Cell Physiol (2008) 295: C557-65 [PMID:18579800] |
| HCN2 in Mouse [GtoPdb: 401] [UniProtKB: O88703] | ||||||||
| GtoPdb | - | - | 3.2 | pIC50 | - | - | - | Am J Physiol, Cell Physiol (2008) 295: C557-65 [PMID:18579800] |
| Kir1.1 in Rat [GtoPdb: 429] [UniProtKB: P35560] | ||||||||
| GtoPdb | - | - | 2.2 | pKi | 6000000 | nM | Ki | J Am Soc Nephrol (2010) 21: 2109-16 [PMID:21030597] |
| GtoPdb | - | - | 2.3 | pKi | 5000000 | nM | Ki |
J Am Soc Nephrol (2010) 21: 2109-16 [PMID:21030597]; J Physiol (Lond.) (1994) 476: 399-409 [PMID:8057249] |
| Kir2.1 in Mouse [GtoPdb: 430] [UniProtKB: P35561] | ||||||||
| GtoPdb | - | - | 4.8 | pKd | 17100 | nM | Kd | Neuron (1995) 14: 1047-54 [PMID:7748552] |
| Kir2.2 in Human [GtoPdb: 431] [UniProtKB: Q14500] | ||||||||
| GtoPdb | - | - | 4.96 | pIC50 | 11000 | nM | IC50 | J Physiol (Lond.) (1996) 493 ( Pt 1): 143-56 [PMID:8735700] |
| Kir2.3 in Human [GtoPdb: 432] [UniProtKB: P48050] | ||||||||
| GtoPdb | - | - | 5 | pKd | 10000 | nM | Kd | Nature (1994) 372: 366-9 [PMID:7969496] |
| TRPC5 in Rat [GtoPdb: 490] | ||||||||
| GtoPdb | - | - | 3.34 | pIC50 | - | - | - | J Neurosci (2005) 25: 1234-9 [PMID:15689561] |
| TRPM3 in Mouse [GtoPdb: 495] | ||||||||
| GtoPdb | - | - | 2 | pIC50 | - | - | - | J Biol Chem (2005) 280: 22540-8 [PMID:15824111] |
| TRPM6 in Human [GtoPdb: 498] [UniProtKB: Q9BX84] | ||||||||
| GtoPdb | - | - | 3.3 | pIC50 | - | - | - | J Biol Chem (2004) 279: 19-25 [PMID:14576148] |
| GtoPdb | - | - | 6 | pIC50 | 1100 | nM | IC50 | |
| TRPM7 in Mouse [GtoPdb: 499] [UniProtKB: Q923J1] | ||||||||
| GtoPdb | - | - | 2.49 | pIC50 | 3200000 | nM | IC50 | Nature (2001) 411: 590-5 [PMID:11385574] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
