Audien   Click here for help

GtoPdb Ligand ID: 10189

Compound class: Inorganic
Comment: Audien is a gold (Au)-containing compound that was designed as a potential antitumor agent [2]. In this reference it is described as Au(dien)Cl]Cl2, where dien = diethylentriamine. It has been shown to act as an inhibitor of aquaglyceroporin AQP3 [1].
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Selectivity at ion channels
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
AQP3 Hs Inhibitor - 4.8 pIC50 - 1
pIC50 4.8 (IC50 1.7x10-5 M) [1]