Ligand id: 10222

Name: TAK-448

Structure and Physico-chemical Properties

2D Structure
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Bioactivity Comments
Subcutaneously delivered TAK-448 suppresses testosterone in rats [2].
Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
kisspeptin receptor Hs Agonist Agonist 8.3 pEC50 - 2
pEC50 8.3 (EC50 5.2x10-9 M) [2]