Synonyms: WX-081
Compound class:
Synthetic organic
Comment: Sudapyridine (WX-081) is the lead from a novel diarylpyridine series with antimycobacterial activity and an analogue of bedaquiline [1,3]. Sudapyridine has advanced to clinical evaluation for the treatment of tuberculosis.
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Bioactivity Comments |
The MIC for antimycobacterial activity against Mycobacterium tuberculosis H37Rv is 0.070 μg/ml in vitro [3]. |