|
|
|
D3 receptor
|
|
|
Rn |
Agonist |
Full agonist |
7.3 – 7.8 |
pKi |
- |
1,10 |
|
⤷ |
pKi
7.3 – 7.8
[1,10]
|
D4 receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.5 |
pKi |
- |
4,7,11 |
|
⤷ |
pKi
7.5
[4,7,11]
|
D3 receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.4 – 8.0 |
pKi |
- |
1,3,5,7-11 |
|
⤷ |
pKi
6.4 – 8.0
(Ki 3.98x10-7 – 1x10-8 M)
[1,3,5,7-11]
|
D2 receptor
|
|
|
Hs |
Agonist |
Full agonist |
4.9 – 7.7 |
pKi |
- |
1,3,7,9-11 |
|
⤷ |
pKi
4.9 – 7.7
[1,3,7,9-11]
|
5-HT1A receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.8 |
pKi |
- |
6 |
|
⤷ |
pKi
5.8
[6]
|
5-HT2B receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.0 – 6.5 |
pKi |
- |
2,4 |
|
⤷ |
pKi
5.0 – 6.5
[2,4]
|
5-HT2A receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.0 – 5.5 |
pKi |
- |
2,4 |
|
⤷ |
pKi
5.0 – 5.5
[2,4]
|
5-HT2C receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.0 – 5.5 |
pKi |
- |
2,4 |
|
⤷ |
pKi
5.0 – 5.5
[2,4]
|
D2 receptor
|
|
|
Rn |
Agonist |
Full agonist |
5.2 |
pKi |
- |
10 |
|
⤷ |
pKi
5.2
[10]
|
|