NC 4-28B   Click here for help

GtoPdb Ligand ID: 2017

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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 8.4 pKi - 2
pKi 8.4 [2]
SST3 receptor Hs Agonist Full agonist 8.0 pKi - 2
pKi 8.0 [2]
SST1 receptor Hs Agonist Full agonist 7.4 pKi - 2
pKi 7.4 [2]
SST2 receptor Mm Agonist Full agonist 10.0 – 11.7 pIC50 - 1,3
pIC50 10.0 – 11.7 [1,3]
SST3 receptor Mm Agonist Full agonist 7.0 pIC50 - 3
pIC50 7.0 [3]