BIM 23030   

GtoPdb Ligand ID: 2034

Comment: Cyclic peptide
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 7.7 – 7.9 pKi - 3-5
pKi 7.7 – 7.9 [3-5]
SST5 receptor Mm Agonist Full agonist 7.1 – 8.0 pKi - 1
pKi 7.1 – 8.0 [1]
SST3 receptor Hs Agonist Full agonist 7.2 – 7.8 pKi - 3,5
pKi 7.2 – 7.8 [3,5]
SST5 receptor Hs Agonist Full agonist 5.6 – 7.4 pKi - 5
pKi 5.6 – 7.4 [5]
SST2 receptor Mm Agonist Full agonist 8.2 pIC50 - 2
pIC50 8.2 [2]