BIM 23068   

GtoPdb Ligand ID: 2040

Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 8.8 pKi - 2
pKi 8.8 [2]
SST3 receptor Hs Agonist Full agonist 8.8 pKi - 2
pKi 8.8 [2]
SST3 receptor Rn Agonist Full agonist 8.4 pKi - 1
pKi 8.4 [1]
SST4 receptor Hs Agonist Full agonist 8.0 pKi - 2
pKi 8.0 [2]
SST2 receptor Mm Agonist Full agonist 9.8 pIC50 - 3
pIC50 9.8 [3]
SST3 receptor Mm Agonist Full agonist 9.1 pIC50 - 3
pIC50 9.1 [3]