|
|
|
5-HT2C receptor
|
|
|
Rn |
Antagonist |
Inverse agonist |
9.2 |
pKi |
- |
6 |
|
⤷ |
pKi
9.2
[6]
|
5-HT2C receptor
|
|
|
Hs |
Antagonist |
Inverse agonist |
8.7 – 9.3 |
pKi |
- |
5,9,11 |
|
⤷ |
pKi
8.7 – 9.3
[5,9,11]
|
5-HT2B receptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.5 – 8.8 |
pKi |
- |
9,11,19 |
|
⤷ |
pKi
8.5 – 8.8
[9,11,19]
|
5-HT2A receptor
|
|
|
Rn |
Antagonist |
Antagonist |
8.6 |
pKi |
- |
8 |
|
⤷ |
pKi
8.6
[8]
|
5-HT7 receptor
|
|
|
Rn |
Antagonist |
Antagonist |
7.7 – 8.2 |
pKi |
- |
15 |
|
⤷ |
pKi
7.7 – 8.2
[15]
|
5-HT7 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.5 – 8.2 |
pKi |
- |
1,7,12,17 |
|
⤷ |
pKi
7.5 – 8.2
[1,7,12,17]
|
5-HT7 receptor
|
|
|
Mm |
Antagonist |
Antagonist |
7.6 |
pKi |
- |
14 |
|
⤷ |
pKi
7.6
[14]
|
5-HT2B receptor
|
|
|
Rn |
Antagonist |
Antagonist |
7.4 |
pKi |
- |
18 |
|
⤷ |
pKi
7.4
[18]
|
5-HT2A receptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.0 – 7.5 |
pKi |
- |
9,16 |
|
⤷ |
pKi
7.0 – 7.5
[9,16]
|
5-HT6 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
5.4 – 5.7 |
pKi |
- |
2,4,10 |
|
⤷ |
pKi
5.4 – 5.7
[2,4,10]
|
5-HT6 receptor
|
|
|
Rn |
Antagonist |
Antagonist |
5.1 – 5.8 |
pKi |
- |
3-4,13 |
|
⤷ |
pKi
5.1 – 5.8
[3-4,13]
|
|