gastric inhibitory polypeptide

Ligand id: 3542

Name: gastric inhibitory polypeptide

Abbreviated name: GIP

Species: Human

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View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Natural/Endogenous Targets
GIP receptor
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
GIP receptor Hs Agonist Full agonist 8.7 pKd - 3
pKd 8.7 [3]
GIP receptor Hs Agonist Agonist 9.1 pKi - 2
pKi 9.1 (Ki 7.5x10-10 M) [2]
GIP receptor Rn Agonist Full agonist 8.6 pIC50 - 1
pIC50 8.6 [1]
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