gastric inhibitory polypeptide   

GtoPdb Ligand ID: 3542

Abbreviated name: GIP
Synonyms: GIP(1-42)
Comment: Human GIP differs from mouse GIP at residues 18 (Histidine), 30 (Lysine) and 34 (Asparagine) and from rat at residues 18 and 40.
Species: Human
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Natural/Endogenous Targets
Target
GIP receptor
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
GIP receptor Hs Agonist Full agonist 8.7 pKd - 3
pKd 8.7 [3]
GIP receptor Hs Agonist Agonist 9.1 pKi - 2
pKi 9.1 (Ki 7.5x10-10 M) [2]
GIP receptor Rn Agonist Full agonist 8.6 pIC50 - 1
pIC50 8.6 [1]
Ligand mentioned in the following text fields