|
|
|
GAL1 receptor
|
|
|
Mm |
Agonist |
Full agonist |
9.3 – 10.3 |
pKi |
- |
11,20 |
|
⤷ |
pKi
9.3 – 10.3
(Ki 4.6x10-10 – 4.7x10-11 M)
[11,20]
|
GAL1 receptor
|
|
|
Rn |
Agonist |
Full agonist |
9.0 – 10.1 |
pKi |
- |
4,14,17-19 |
|
⤷ |
pKi
9.0 – 10.1
(Ki 1x10-9 – 8x10-11 M)
[4,14,17-19]
|
GAL1 receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.8 – 10.1 |
pKi |
- |
2,7-9,12-13,15 |
|
⤷ |
pKi
8.8 – 10.1
(Ki 1.75x10-9 – 8x10-11 M)
[2,7-9,12-13,15]
|
GAL2 receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.3 – 9.3 |
pKi |
- |
8,11,14,17-19 |
|
⤷ |
pKi
8.3 – 9.3
(Ki 5.6x10-9 – 5.6x10-10 M)
[8,11,14,17-19]
|
GAL2 receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.5 – 8.8 |
pKi |
- |
1-2,9,12-13,15 |
|
⤷ |
pKi
8.5 – 8.8
(Ki 2.98x10-9 – 1.54x10-9 M)
[1-2,9,12-13,15]
|
GAL3 receptor
|
|
|
Rn |
Agonist |
Partial agonist |
8.1 – 8.8 |
pKi |
- |
8,14,17,19 |
|
⤷ |
pKi
8.1 – 8.8
(Ki 7.4x10-9 – 1.47x10-9 M)
[8,14,17,19]
|
GAL2 receptor
|
|
|
Mm |
Agonist |
Full agonist |
8.4 |
pKi |
- |
11 |
|
⤷ |
pKi
8.4
(Ki 3.9x10-9 M)
[11]
|
GAL3 receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.9 – 8.4 |
pKi |
- |
2,12-14,16 |
|
⤷ |
pKi
7.9 – 8.4
(Ki 1.23x10-8 – 4.49x10-9 M)
[2,12-14,16]
|
GAL1 receptor
|
|
|
Rn |
Agonist |
Full agonist |
9.8 |
pEC50 |
- |
10 |
|
⤷ |
pEC50
9.8
(EC50 1.6x10-10 M)
[10]
|
GAL2 receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.3 |
pEC50 |
- |
10 |
|
⤷ |
pEC50
8.3
(EC50 5.2x10-9 M)
[10]
|
GAL1 receptor
|
|
|
Hs |
Agonist |
Full agonist |
9.9 |
pIC50 |
- |
5 |
|
⤷ |
pIC50
9.9
(IC50 1.3x10-10 M)
[5]
|
GAL1 receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.9 – 10.0 |
pIC50 |
- |
3,10 |
|
⤷ |
pIC50
8.9 – 10.0
(IC50 1.4x10-9 – 9.7x10-11 M)
[3,10]
|
GAL2 receptor
|
|
|
Rn |
Agonist |
Full agonist |
8.7 – 9.3 |
pIC50 |
- |
3,6,10 |
|
⤷ |
pIC50
8.7 – 9.3
(IC50 1.9x10-9 – 4.8x10-10 M)
[3,6,10]
|
GAL2 receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.9 – 9.5 |
pIC50 |
- |
2,5 |
|
⤷ |
pIC50
9.5
(IC50 3.4x10-10 M)
[5]
pIC50
7.9 – 9.1
(IC50 1.175x10-8 – 7.6x10-10 M)
[2,5]
|
GAL3 receptor
|
|
|
Rn |
Agonist |
Full agonist |
7.0 |
pIC50 |
- |
3 |
|
⤷ |
pIC50
7.0
(IC50 1.084x10-7 M)
[3]
|
|