[D-Phe6, Leu13, Cpa14,ψ13-14]bombesin-(6-14)   

GtoPdb Ligand ID: 3840

Synonyms: [D-Phe6,Cpa14,ψ13-14]bombesin6-14 | [D-Phe6,Leu13,Cpa14,ψ13-14]bombesin-(6-14) | analogue #7 [PMID: 19463875]
Comment: Synthetic analogue of bombesin [1].
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
BB2 receptor Hs Antagonist Antagonist 9.8 pKi - 1
pKi 9.8 [1]
BB2 receptor Rn Antagonist Antagonist 7.4 pKi - 2
pKi 7.4 (Ki 4.2x10-8 M) [2]
BB2 receptor Hs Antagonist Antagonist 8.9 – 8.9 pIC50 - 1
pIC50 8.9 – 8.9 (IC50 1.35x10-9 – 1.23x10-9 M) [1]
BB1 receptor Hs Antagonist Antagonist <5.0 pIC50 - 1
pIC50 <5.0 (IC50 >1x10-5 M) [1]