Ligand id: 2322

Name: chlorzoxazone

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Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 1
Hydrogen bond donors 1
Rotatable bonds 0
Topological polar surface area 46
Molecular weight 168.99
XLogP 1.61
No. Lipinski's rules broken 0

Molecular properties generated using the CDK

No information available.
Summary of Clinical Use
Used to treat painful musculoskeletal conditions.
Mechanism Of Action and Pharmacodynamic Effects
CHEMBL lists Intermediate conductance calcium-activated potassium channel protein 4 (gene symbol KCNN4) as the target of this drug, but it also thought that inhibition of histamine release from mast cells plays a part in its mechanism of action.