[D-Phe6,β-Ala11,Phe13,Nle14]bombesin-(6-14)   Click here for help

GtoPdb Ligand ID: 632

Synonyms: [D-Phe6,β-Ala11,Phe13,Nle14]bombesin(6-14)
Comment: Synthetic analogue of bombesin
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1. Hoppenz P, Els-Heindl S, Beck-Sickinger AG. (2019)
Identification and stabilization of a highly selective gastrin-releasing peptide receptor agonist.
J Pept Sci, 25 (12): e3224. [PMID:31743956]
2. Mantey SA, Weber HC, Sainz E, Akeson M, Ryan RR, Pradhan TK, Searles RP, Spindel ER, Battey JF, Coy DH et al.. (1997)
Discovery of a high affinity radioligand for the human orphan receptor, bombesin receptor subtype 3, which demonstrates that it has a unique pharmacology compared with other mammalian bombesin receptors.
J Biol Chem, 272 (41): 26062-71. [PMID:9325344]
3. Ryan RR, Katsuno T, Mantey SA, Pradhan TK, Weber HC, Coy DH, Battey JF, Jensen RT. (1999)
Comparative pharmacology of the nonpeptide neuromedin B receptor antagonist PD 168368.
J Pharmacol Exp Ther, 290 (3): 1202-11. [PMID:10454496]
4. Uehara H, Gonz├ílez N, Sancho V, Mantey SA, Nuche-Berenguer B, Pradhan T, Coy DH, Jensen RT. (2011)
Pharmacology and selectivity of various natural and synthetic bombesin related peptide agonists for human and rat bombesin receptors differs.
Peptides, 32 (8): 1685-99. [PMID:21729729]