ChEMBL ligand: CHEMBL148319
Peroxisome proliferator-activated receptor-α/Peroxisome proliferator-activated receptor alpha in Human [ChEMBL: CHEMBL239] [GtoPdb: 593] [UniProtKB: Q07869] There should be some charts here, you may need to enable JavaScript!
Peroxisome proliferator-activated receptor-β/δ/Peroxisome proliferator-activated receptor delta in Human [ChEMBL: CHEMBL3979] [GtoPdb: 594] [UniProtKB: Q03181] There should be some charts here, you may need to enable JavaScript!
Peroxisome proliferator-activated receptor-γ/Peroxisome proliferator-activated receptor gamma in Human [ChEMBL: CHEMBL235] [GtoPdb: 595] [UniProtKB: P37231] There should be some charts here, you may need to enable JavaScript!
DP1 receptor in Human [GtoPdb: 338] [UniProtKB: Q13258] There should be some charts here, you may need to enable JavaScript!
EP1 receptor in Human [GtoPdb: 340] [UniProtKB: P34995] There should be some charts here, you may need to enable JavaScript!
EP2 receptor in Human [GtoPdb: 341] [UniProtKB: P43116] EP2 receptor in Mouse [GtoPdb: 341] [UniProtKB: Q62053] There should be some charts here, you may need to enable JavaScript!
EP3 receptor in Human [GtoPdb: 342] [UniProtKB: P43115] EP3 receptor in Mouse [GtoPdb: 342] [UniProtKB: P30557] There should be some charts here, you may need to enable JavaScript!
EP4 receptor in Human [GtoPdb: 343] [UniProtKB: P35408] EP4 receptor in Mouse [GtoPdb: 343] [UniProtKB: P32240] There should be some charts here, you may need to enable JavaScript!
FP receptor in Human [GtoPdb: 344] [UniProtKB: P43088] FP receptor in Mouse [GtoPdb: 344] [UniProtKB: P43117] There should be some charts here, you may need to enable JavaScript!
IP receptor in Human [GtoPdb: 345] [UniProtKB: P43119] IP receptor in Mouse [GtoPdb: 345] [UniProtKB: P43252] There should be some charts here, you may need to enable JavaScript!
TP receptor in Human [GtoPdb: 346] [UniProtKB: P21731] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
Peroxisome proliferator-activated receptor-α/Peroxisome proliferator-activated receptor alpha in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL239] [GtoPdb: 593] [UniProtKB: Q07869]
ChEMBL	In vitro transactivation of human Peroxisome proliferator activated receptor alpha (hPPARalpha)	B	6.02	pEC50	960	nM	EC50	J Med Chem (2003) 46: 4883-4894 [PMID:14584939]
ChEMBL	In vitro transactivation using receptor transactivation assay against hPPAR alpha	F	6.47	pEC50	340	nM	EC50	J Med Chem (2002) 45: 789-804 [PMID:11831892]
Peroxisome proliferator-activated receptor-β/δ/Peroxisome proliferator-activated receptor delta in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3979] [GtoPdb: 594] [UniProtKB: Q03181]
ChEMBL	In vitro transcriptional activation of hPPAR delta	F	5.62	pEC50	2410	nM	EC50	J Med Chem (2002) 45: 789-804 [PMID:11831892]
ChEMBL	In vitro transactivation of human Peroxisome proliferator activated receptor delta (hPPARdelta)	B	5.73	pEC50	1880	nM	EC50	J Med Chem (2003) 46: 4883-4894 [PMID:14584939]
Peroxisome proliferator-activated receptor-γ/Peroxisome proliferator-activated receptor gamma in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL235] [GtoPdb: 595] [UniProtKB: P37231]
ChEMBL	In vitro transactivation of human Peroxisome proliferator activated receptor gamma	B	5.1	pEC50	7910	nM	EC50	J Med Chem (2003) 46: 4883-4894 [PMID:14584939]
DP1 receptor in Human [GtoPdb: 338] [UniProtKB: Q13258]
GtoPdb	-	-	6.9	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
EP1 receptor in Human [GtoPdb: 340] [UniProtKB: P34995]
GtoPdb	-	-	7.6	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
EP2 receptor in Human [GtoPdb: 341] [UniProtKB: P43116]
GtoPdb	-	-	6	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
EP2 receptor in Mouse [GtoPdb: 341] [UniProtKB: Q62053]
GtoPdb	-	-	5.8	pKi	-	-	-	Br J Pharmacol (1997) 122: 217-24 [PMID:9313928]
EP3 receptor in Human [GtoPdb: 342] [UniProtKB: P43115]
GtoPdb	-	-	7.85	pKi	14	nM	Ki	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
EP3 receptor in Mouse [GtoPdb: 342] [UniProtKB: P30557]
GtoPdb	-	-	7.51	pKi	31	nM	Ki	Br J Pharmacol (1997) 122: 217-24 [PMID:9313928]
EP4 receptor in Human [GtoPdb: 343] [UniProtKB: P35408]
GtoPdb	-	-	6.5	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
EP4 receptor in Mouse [GtoPdb: 343] [UniProtKB: P32240]
GtoPdb	-	-	5.6	pKi	-	-	-	Br J Pharmacol (1997) 122: 217-24 [PMID:9313928]
FP receptor in Human [GtoPdb: 344] [UniProtKB: P43088]
GtoPdb	-	-	6.5	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
FP receptor in Mouse [GtoPdb: 344] [UniProtKB: P43117]
GtoPdb	-	-	5.9	pKi	-	-	-	Br J Pharmacol (1997) 122: 217-24 [PMID:9313928]
IP receptor in Human [GtoPdb: 345] [UniProtKB: P43119]
GtoPdb	-	-	6.6	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]
IP receptor in Mouse [GtoPdb: 345] [UniProtKB: P43252]
GtoPdb	-	-	7	pKi	-	-	-	Br J Pharmacol (1997) 122: 217-24 [PMID:9313928]
TP receptor in Human [GtoPdb: 346] [UniProtKB: P21731]
GtoPdb	-	-	4.7	pKi	-	-	-	Biochim Biophys Acta (2000) 1483: 285-93 [PMID:10634944]

ChEMBL data shown on this page come from version 32:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]