|
|
|
5-HT2B receptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.4 – 9.0 |
pKi |
- |
6,11 |
|
⤷ |
pKi
8.4 – 9.0
[6,11]
|
5-HT2B receptor
|
|
|
Rn |
Antagonist |
Antagonist |
8.3 – 8.4 |
pKi |
- |
6,10 |
|
⤷ |
pKi
8.3 – 8.4
[6,10]
|
5-HT1D receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.1 – 8.2 |
pKi |
- |
5,12 |
|
⤷ |
pKi
8.1 – 8.2
[5,12]
|
5-HT1A receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.0 |
pKi |
- |
5 |
|
⤷ |
pKi
8.0
[5]
|
5-HT1B receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.7 – 7.9 |
pKi |
- |
5,8,12 |
|
⤷ |
pKi
7.7 – 7.9
[5,8,12]
|
5-HT7 receptor
|
|
|
Rn |
Agonist |
Full agonist |
7.5 – 7.7 |
pKi |
- |
9 |
|
⤷ |
pKi
7.5 – 7.7
[9]
|
5-HT1F receptor
|
|
|
Hs |
Antagonist |
Antagonist |
7.3 |
pKi |
- |
1-2 |
|
⤷ |
pKi
7.3
[1-2]
|
5-HT7 receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.1 |
pKi |
- |
4 |
|
⤷ |
pKi
7.1
[4]
|
5-HT6 receptor
|
|
|
Rn |
Agonist |
Full agonist |
7.0 |
pKi |
- |
7 |
|
⤷ |
pKi
7.0
[7]
|
5-ht1e receptor
|
|
|
Hs |
Antagonist |
Antagonist |
6.7 – 7.0 |
pKi |
- |
2-3,8 |
|
⤷ |
pKi
6.7 – 7.0
[2-3,8]
|
|