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Synonyms: GSK 962040 | GSK962040
Compound class: Synthetic organic
Comment: Camicinal is a motilin receptor agonist.
Ligand Activity Visualisation Charts
These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.✖
1. Barshop K, Kuo B. (2015)
The investigational drug camicinal for the treatment of gastroparesis.
Expert Opin Investig Drugs, 24 (1): 133-140. [PMID:25341626]
2. Chapman MJ, Deane AM, O'Connor SL, Nguyen NQ, Fraser RJ, Richards DB, Hacquoil KE, Vasist Johnson LS, Barton ME, Dukes GE. (2016)
The effect of camicinal (GSK962040), a motilin agonist, on gastric emptying and glucose absorption in feed-intolerant critically ill patients: a randomized, blinded, placebo-controlled, clinical trial.
Crit Care, 20 (1): 232. [PMID:27476581]
3. Peeters TL. (2015)
Gastrointestinal hormones and gut motility.
Curr Opin Endocrinol Diabetes Obes, 22 (1): 9-13. [PMID:25517024]
4. Sanger GJ, Westaway SM, Barnes AA, Macpherson DT, Muir AI, Jarvie EM, Bolton VN, Cellek S, Näslund E, Hellström PM et al.. (2009)
GSK962040: a small molecule, selective motilin receptor agonist, effective as a stimulant of human and rabbit gastrointestinal motility.
Neurogastroenterol Motil, 21 (6): 657-64, e30-1. [PMID:19374732]