BIM 23052   

GtoPdb Ligand ID: 2004

Synonyms: BIM-23052 | BIM23052 | DC-(23-99)
Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST3 receptor Hs Agonist Full agonist 8.4 – 9.7 pKi - 1,4,6
pKi 8.4 – 9.7 [1,4,6]
SST5 receptor Rn Agonist Full agonist 8.6 pKi - 2
pKi 8.6 [2]
SST3 receptor Rn Agonist Full agonist 8.5 pKi - 2
pKi 8.5 [2]
SST5 receptor Hs Agonist Full agonist 7.4 – 9.6 pKi - 2,4-6
pKi 7.4 – 9.6 [2,4-6]
SST2 receptor Hs Agonist Full agonist 8.1 – 8.8 pKi - 1,4-6
pKi 8.1 – 8.8 [1,4-6]
SST1 receptor Hs Agonist Full agonist 8.2 – 8.6 pKi - 1,4,6
pKi 8.2 – 8.6 [1,4,6]
SST4 receptor Hs Agonist Full agonist 8.2 – 8.6 pKi - 4
pKi 8.2 – 8.6 [4]
SST3 receptor Mm Agonist Full agonist 9.4 pIC50 - 3
pIC50 9.4 [3]
SST4 receptor Rn Agonist Full agonist 8.1 pIC50 - 7
pIC50 8.1 [7]