BIM 23056   Click here for help

GtoPdb Ligand ID: 2036

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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST5 receptor Mm Agonist Full agonist 7.5 – 7.9 pKd - 2
pKd 7.5 – 7.9 [2]
SST5 receptor Hs Antagonist Antagonist 7.4 – 8.3 pKi -
pKi 7.4 – 8.3
SST5 receptor Hs Agonist Full agonist 6.7 – 8.3 pKi - 3-4,6-8
pKi 6.7 – 8.3 [3-4,6-8]
SST3 receptor Hs Agonist Full agonist 6.9 – 7.2 pKi - 6,8
pKi 6.9 – 7.2 [6,8]
SST2 receptor Hs Agonist Full agonist 6.2 – 6.7 pKi - 1,6-8
pKi 6.2 – 6.7 [1,6-8]
SST5 receptor Rn Agonist Full agonist 6.3 pKi - 3
pKi 6.3 [3]
SST3 receptor Mm Agonist Full agonist 10.7 pIC50 - 5
pIC50 10.7 [5]
SST3 receptor Rn Agonist Full agonist 6.5 pIC50 - 9
pIC50 6.5 [9]