BIM 23056

Ligand id: 2036

Name: BIM 23056

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST5 receptor Mm Agonist Full agonist 7.5 – 7.9 pKd - 2
pKd 7.5 – 7.9 [2]
SST5 receptor Hs Antagonist Antagonist 7.4 – 8.3 pKi -
pKi 7.4 – 8.3
SST5 receptor Hs Agonist Full agonist 6.7 – 8.3 pKi - 3-4,6-8
pKi 6.7 – 8.3 [3-4,6-8]
SST3 receptor Hs Agonist Full agonist 6.9 – 7.2 pKi - 6,8
pKi 6.9 – 7.2 [6,8]
SST2 receptor Hs Agonist Full agonist 6.2 – 6.7 pKi - 1,6-8
pKi 6.2 – 6.7 [1,6-8]
SST5 receptor Rn Agonist Full agonist 6.3 pKi - 3
pKi 6.3 [3]
SST3 receptor Mm Agonist Full agonist 10.7 pIC50 - 5
pIC50 10.7 [5]
SST3 receptor Rn Agonist Full agonist 6.5 pIC50 - 9
pIC50 6.5 [9]