[125I]Tyr10-CST14   Click here for help

GtoPdb Ligand ID: 2024

Synonyms: [125I]-[Tyr10]CST-14 | [125I]Tyr10-cortistatin14
 Ligand is labelled  Ligand is radioactive
Compound class: Peptide
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Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST5 receptor Hs Agonist Full agonist 10.3 pKd - 2-3
pKd 10.3 [2-3]
SST5 receptor Mm Agonist Full agonist 10.2 pKd - 1
pKd 10.2 [1]
SST3 receptor Hs Agonist Full agonist 10.1 pKd - 2-3
pKd 10.1 [2-3]
SST1 receptor Hs Agonist Full agonist 10.0 pKd - 2-3
pKd 10.0 [2-3]
SST2 receptor Hs Agonist Full agonist 9.4 pKd - 2-3
pKd 9.4 [2-3]
SST4 receptor Hs Agonist Full agonist 9.4 pKd - 3
pKd 9.4 [3]
Ligand mentioned in the following text fields