Available chemical structures for TRPM8 channel blockers

PBMC
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Targets
TRPM8
M8-B
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Targets
TRPM8
PF-05105679
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Targets
TRPM8
BCTC
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Targets
TRPM8; TRPV1
scutellarein
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Targets
TAS2R39; CoV Non-structural protein 13; TRPM8
cannabidiol
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Targets
GPR55; CB1 receptor; Nav1.1; Nav1.2; Nav1.3; Nav1.4; Nav1.5; Nav1.6; Nav1.7; Nav1.8; TRPA1; TRPM8; TRPV2; TRPV3
thio-BCTC
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Targets
TRPM8
2-APB
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Targets
TRPC1; TRPC2; TRPC3; TRPC4; TRPC5; TRPC6; TRPC7; TRPM2; TRPM3; TRPM6; TRPM7; TRPM8; TRPV1; TRPV2; TRPV3... click on ligand to see complete list
capsazepine
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Targets
TRPM8; TRPV1
5-benzyloxytryptamine
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Targets
5-HT6 receptor; TRPM8
linoleic acid
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Targets
FFA1 receptor; FFA4 receptor; Hepatocyte nuclear factor-4-α; Kv2.1; K2P10.1; Peroxisome proliferator-activated receptor-γ; TRPM8; cellular retinoic acid binding protein 1; fatty acid binding protein 1; fatty acid binding protein 2; fatty acid binding protein 3; fatty acid binding protein 4; retinol binding protein 2
clotrimazole
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Targets
Constitutive androstane receptor; KCa1.1; KCa3.1; Pregnane X receptor; TRPM2; TRPM3; TRPM4; TRPM8
anandamide
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Targets
GPR119; GPR18; GPR55; CB1 receptor; CB2 receptor; Cav3.2; Cav3.3; Glycine Receptor (All subtypes); Kv1.2; K2P3.1; K2P9.1; TRPM8; TRPV1; glycine receptor α1 subunit; monoacylglycerol lipase... click on ligand to see complete list
Δ9-tetrahydrocannabinol
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Targets
GPR18; GPR55; CB1 receptor; CB2 receptor; TRPA1; TRPM8; TRPV2; glycine receptor α1 subunit; glycine receptor α2 subunit; glycine receptor α3 subunit
ACAA
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Targets
TRPC3; TRPC6; TRPM2; TRPM8
AMTB
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Targets
TRPM8
NADA
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Targets
TRPM8; TRPV1

Please note that chemical structures may not be available for all channel blockers at this target. For more details please email us.