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The IUPHAR/BPS Guide to PHARMACOLOGY complete ligand list

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Synthetic, semi-synthetic and natural peptides encoded in genomes other than human, rat and mouse (including oligopeptides and cyclic peptides).

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Ligand name ID Synonyms
A Back to top
A-71378 894 A 71378, A71378
A-71623 858 A 71623, A71623, L-phenylalaninamide
A-71915 4856 A 71915, A71915, H-3048
A8Δ71-73 5780
abaloparatide Approved drug 8299 BA058, Tymlos®
abarelix Approved drug 1188 Plenaxis®, PPI 149, R 3827
A(4-24)(B7-24)H2 8346 A(4-24)(B7-24)H2 relaxin
A(4-24)(B7-24)H2 chain A 8347 A(4-24)H2 relaxin
A(4-24)(B7-24)H2 chain B 8348 (B7-24)H2 relaxin
abicipar pegol 8371 AGN-150998, MP0112
ABS-201 5308 ABS 201, ABS201, HPI-201, HPI201, KK13
ABS-212 5307 ABS 212, ABS212
Abz-Ser-Pro-Tyr(NO2)-OH 5132 o-aminobenzoyl-Ser-Pro-Tyr(NO2)-OH, TBC5182
AC-178,335 2065 AC 178335
AC187 689 AC 187, AC-187, acetyl-(Asn30,Tyr32)-calcitonin8-32, salmon calcitonin (8-32) reduced
Ac-c[Cys-Glu-His-D-Phe-Arg-Trp-D-Cys]-Pro-Pro-Lys-Asp-NH2 1342
[Ac-D-2Nal1,D4CPA2,D-3Pal3,6,Leu8, D-Ala10]GnRH-II 5583
Ac-GRP-(20-26)-methylester 625 N-acetyl-GRP-(20-26)-ethylester
[Ac-His1]PACAP-27 2263 [Ac-His1]pituitary adenylate cyclase activating polypeptide-27
[125I][Ac-His1]PACAP-27 Ligand is labelled Ligand is radioactive 2260 [125I]-[Ac-His1]pituitary adenylate cyclase activating polypeptide-27
Ac-hMCH-(6-16)-NH2 1290 hAc-MCH(6-16)-NH2, human Ac-MCH6-16-NH2
A(Δ10/15C)INSL3 8332
aclerastide 8300 DSC-127, DSC127, NorLeu3-A(1-7)
Ac-Lys-[MeAla6,Leu8,des-Arg9]bradykinin 651 N-acetylated-[Lys,MeAla6,Leu8,des-Arg9]bradykinin, Ac-[MeAla6,Leu8,des-Arg9]kallidin
AcPhe-Orn-Pro-D-Cha-Trp-Arg 3853 AcF[OP-D-Cha-Wr]
Ac-Phe-Trp-Ala-His(τBZL)-Nip-Gly-Arg-NH2 6191
Ac-RHYPLWR 8380
Ac-RYYRIK-NH2 1679
Ac-RYYRWK-NH2 1680
Ac-SDKP Immunopharmacology Ligand 10060 goralatide, seraspenide
A(C10/15S)INSL3 8331
ACTH-(11-24) 1332 ACTH (11-24), adrenocorticotropic hormone (11-24)
ACTH-(1-24) 1330 ACTH (1-24), adrenocorticotropic hormone (1-24)
[125I]ACTH-(1-24) Ligand is labelled Ligand is radioactive 3767 [125I]-ACTH(1-24), [125I]-adrenocorticotropin(1-24)
[Ac-Tyr1, D-Arg2]GHRH-(1-29)-NH2 (human) 1125
AF12198 Immunopharmacology Ligand 4861 AF 12198, AF-12198
A(4-24)(F23A)H2 8349
afamelanotide Approved drug 1324 α-NDP-MSH, [Nle4,dPhe7]α-MSH, CUV-1647, CUV1647, NDP-MSH, Scenesse®
AFT-II 2613 neurotoxin-2, Toxin AFII, Toxin AFT-II
ω-agatoxin IIIA 2528 omega-Aga-IIIA, Omega-agatoxin-Aa3a
ω-agatoxin IVA 2529 omega-Aga-IVA, Omega-agatoxin-Aa4a
ω-agatoxin IVB 2530 Omega-agatoxin-Aa4b
A(10-24)INSL3 8330
A(9-26)INSL3 8329
AL-78898A Immunopharmacology Ligand 9219 4(1MeW), POT-4
[Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]PTH-(1-34)-NH2 5573 [Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]-hPTH 1-34-NH2, M-PTH(1-34)
[Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]PTH-(1-21)-NH2 (human) 5575 [Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]hPTH-(1-21)-NH2, [Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]-PTH 1-21-NH2 (human), M-PTH(1-21)
[Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]PTH-(1-28)-NH2 (human) 5574 [Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]-hPTH 1-28-NH2, [Ala1,12,Aib3,Gln10,hArg11,Trp14,Arg19]-PTH 1-28-NH2 (human), M-PTH(1-28)
[Ala1,12,Aib3,Gln10,hArg11,Trp14]PTH-(1-14)-NH2 5576 [Ala1,12,Aib3,Gln10,hArg11,Trp14]-hPTH 1-14-NH2, [Ala1,12,Aib3,Gln10,hArg11,Trp14]-PTH 1-14-NH2 (human), M-PTH(1-14)
[Ala31,Aib32]NPY 1560
[Ala31,Aib32]NPY (pig) 1522
[Ala11, D-Leu15]orexin-B 1700
[Ala6, D-Trp8]galanin-(1-15)-ol 6146
[Ala1,3,11,15]ET-1 3837 [Ala1,3,11,15]endothelin-1
[125I][Ala1,3,11,15]ET-1 Ligand is labelled Ligand is radioactive 3760 [125I]-[Ala1,3,11,15]endothelin-1, [125I][Ala1,3,11,15]endothelin-1
alafosfalin PDB Ligand 9503 alaphosphin
[2Ala]-galparan 6098
β-Ala-Lys-AMCA Ligand is labelled 9501 β-alanyl-lysyl-N-7-amino-4-methylcoumarin-3-acetic acid, Beta-Ala-Lys-N(epsilon)-AMCA
[βAla8]neurokinin A-(4-10) 2112 [βAla8]neurokinin A (4-10)
alarelin 9342
[Ala11,22,28]VIP 2278 [Ala11,22,28]vasoactive intestinal peptide
albiglutide Approved drug 7386 Eperzan®, GSK716155, Tanzeum®
albutensin A 10226
alglucosidase alfa Approved drug 7561 Lumizyme®, Myozyme®, rhGAA
ALM201 11485
alpha1-proteinase inhibitor Approved drug 7487 A1AT, A1PI, alpha 1-antitrypsin, Aralast®, Prolastin®, serum trypsin inhibitor
AlprolixTM Approved drug 7373
ALT-803 Immunopharmacology Ligand 9615
alunacedase alfa 11320 APN01, GSK-2586881, GSK2586881, rhsACE2
ALX40-4C 607 ALX 40-4C, N-alpha-acetyl-nona-D-arginine amide acetate
AM3 5635 DOTA-Tyr-cyclo(DAB-Arg-cyclo(Cys-Phe-D-Trp-Lys-Thr-Cys)
AM-6120 Immunopharmacology Ligand 10119 AM6120, peptide 41 [PMID: 30346167]
amanitin 4632 α-amanitin
AMG3054 9587
AM-(22-52) (human) 706 AM (22-52), human adrenomedullin (22-52)
AM-(11-50) (rat) 704 AM (11-50), rat adrenomedullin (11-50)
AM-(20-50) (rat) 705 rat adrenomedullin (20-50)
[125I]AM (rat) Ligand is labelled Ligand is radioactive 3768 [125I]-adrenomedullin, [125I]-AM
anakinra Approved drug Immunopharmacology Ligand 6972 antril, Kineret®
analog 30 [PMID:18543899] 5647
analog 31 [PMID:18543899] 5648
analog 32 [PMID:18543899] 7763
analog 3 [PMID:18543899] 5646
anantin 4866
andexanet alfa Approved drug 7576 Andexxa®, coagulation factor Xa (recombinant), inactivated-zhzo, Ondexxya®, PRT064445, PRT4445, r-antidote
[125I]angiotensin-(1-7) (human, mouse, rat) Ligand is labelled Ligand is radioactive 5578 [125I]ang-(1-7)
[125I]ANP (human) Ligand is labelled Ligand is radioactive 4845 [125I]-ANP
antarelix 1189 D-23234, EP 24332
antisauvagine 931 [dPhe11,His12]Svg(11-40), antisauvagine-30
[125I]antisauvagine Ligand is labelled Ligand is radioactive 930
AP811 4870 AP 811, AP-811
apamin 2311
[125I]apelin-13 Ligand is labelled Ligand is radioactive 602
apelin-13(F13A) 5354
APETx-1 2609 Toxin APETx1
APETx2 4135
apraglutide 10685 CVQ1IAY2G6, FE 203799, FE203799
aprotinin  {Sp: Bovine} Approved drug 6570 basic protease inhibitor (BPI), BPTI, pancreatic trypsin inhibitor, Trasylol®
AR305352 7043
[Arg16]chicken secretin 3293 [R16]chicken secretin
arginine vasotocin 2169 AVT, [Arg8]vasotocin
[Arg14Lys15]N/OFQ 1689 [Arg14Lys15]nociceptin, [Arg14Lys15]nociceptin/orphanin FQ, [Arg14Lys15]orphanin FQ
[Arg19]PTH-(1-34) (human) 1792 [Arg19]-PTH 1-34 (human)
ARL-15849 859 AR-R 15849, ARL 15849XX, FPL 15849
ASIP [90-132 (L89Y)] 1327 agouti-signaling protein [90-132 (L89Y)], agouti-signaling protein[90-132 (L89Y)]
astressin 925
[125I]astressin Ligand is labelled Ligand is radioactive 924
astressin 2B 10335 Astressin2-B, astressin2-B, cyclo(31-34)[DPhe(11),His(12),C(alpha)MeLeu(13,39),Nle(17),Glu(31),Lys(34)]Ac-sauvagine(8-40), peptide 20 [PMID: 12361401]
[Asu7,23']β-ANP-(7-28) 4852 [Asu7,23']-β-ANP7-28
atacicept Immunopharmacology Ligand 9517 TACI-Fc, TACI-Ig
atosiban Approved drug 2213 Antocin®, d[D-Tyr(Et)2,Thr4,Orn8]vasotocin, d[D-Tyr(Et)2,Thr4]OVT, ORF22164, RWJ 22164, Tractocile®
ATX-II 2614 anemonia viridis toxin 2, Sea anemone toxin II (Anemonia sulcata), toxin ATX-II
aTyr 1940 8738 ATYR1940, HRS(1-506), Resolaris
AUNP-12 10117 Aur-012, Aurigene NP-12, Aurigene-012, compound #8 [WO2011161699A3]
Ava3 3855
Ava5 3856
[Ava9,10,Ava14,15]-Ac-hMCH6-16-NH2 1307 compound 30 [PMID:12009900]
aviptadil Approved drug 10891 Invicorp® (aviptadil + phentolamine), Vasoactive intestinal octacosapeptide
[3H]AVP (human, mouse, rat) Ligand is labelled Ligand is radioactive 2175 [3H]arginine vasopressin
AY77 9455 compound 14 [PMID: 26819675]
AYPGKF-NH2 4061 AY-NH2
azapro-3 Immunopharmacology Ligand 9221
 
B Back to top
B-10356 652
B1-27 11459 analog 2 [PMID: 32133341]
B-9430 653 B 9430, B9430
B-9858 654 B 9858, Lys-Lys-[Hyp3, Igl5, D-Igl7, Oic8]des-Arg9-BK
B-9958 655 B9958, des-Arg(9)-BK
barusiban 10890 C4.6,S1-cyclo[N-(3-sulfanylpropanoyl)-D-tryptophyl-L-isoleucyl-L-alloisoleucyl-L-asparaginyl-L-2-aminobutanoyl-N-methyl-L-ornithinol], FE 200 440, FE-200440
BASS antagonist 5644 BASS antagonist Analog 4
BAY 55-9837 2269
BAY86-7548 11260
[125I]BAY 55-9837 Ligand is labelled Ligand is radioactive 2281
BBL-454 895 BBL 454, BBL454
BC-254 896 BC 254, BC254
BC-264 897 BC 264, BC264
Bc-III 2615 major neurotoxin BcIII
[125I]BDNF (human) Ligand is labelled Ligand is radioactive 4846 [125I]-BDNF, [125I]-brain-derived neurotrophic factor
BeKm-1 2610 neurotoxin BeKm-1, potassium channel toxin γ-KTx 2.1
bempegaldesleukin Immunopharmacology Ligand 10659 NKTR-214, NKTR214
BgK 2551 Potassium channel toxin Bgk
[125I]BgK (W5Y / Y26F) Ligand is labelled Ligand is radioactive 2565
(B7-33)H2 9321
[125I]BH-AMY (rat, mouse) Ligand is labelled Ligand is radioactive 3770 [125I]-BH-AMY, [125I]-Bolton Hunter amylin
[125I]BH-MIT1 Ligand is labelled Ligand is radioactive 8522
[125I]BH-NMB (human, mouse, rat) Ligand is labelled Ligand is radioactive 3771 [125I]-BH-NMB, [125I]-Bolton Hunter neuromedin B
[125I]BH-[Sar9,Met(O2)11]SP Ligand is labelled Ligand is radioactive 3769 [125I]-BH-[Sar9,Met(O2)11]SP, [125I]-Bolton Hunter-[Sar9,Met(O2)11]substance P
[3H]BH-[Sar9,Met(O2)11]SP Ligand is labelled Ligand is radioactive 3811 [3H]-Bolton Hunter-[Sar9,Met(O2)11]substance P, [3H]-BH-[Sar9,Met(O2)11]SP
bihelical apoA-I mimetic peptide 5A Immunopharmacology Ligand 9183 5A peptide
BIM 23023 2032
BIM 23027 2033 BIM23027
BIM 23030 2034
BIM 23034 2035 DC 13-212
BIM 23050 2003 BIM-23050
BIM 23052 2004 BIM-23052, BIM23052, DC-(23-99)
BIM 23056 2036
BIM 23058 2068
BIM 23059 2037
BIM 23060 2038
BIM 23066 2039
BIM 23068 2040
BIM 23127 2162
BIM 23197 2041
BIM 23268 2083 BIM23268
BIM 23295 2069
BIM 23313 2084
BIM 23454 2026
BIM 23627 2027 H-5886, MW 1164
BIM28011 3857 [D-Ala2,Ala8,9,15,27,D-Arg29]hGHRH(1-29)NH2, BIM 28011
BIM 28163 1101 BIM-28163
[125I]BIM23027 Ligand is labelled Ligand is radioactive 3772 [125I]-BIM 23027, [125I]-BIM23027
BIO1211 6589 BIO 1211, BIO-1211
bivalirudin Approved drug 6470 Angiomax®
BJP-06-005-3 11401 compound 1 [PMID: 32483379], N-(chloroacetyl)-N-methyl-L-phenylalanyl-L-homoprolyl-L-tryptophyl-L-citrulline ethyl ester
[3H]BK (human, mouse, rat) Ligand is labelled Ligand is radioactive 3812 [3H]-BK, [3H]-bradykinin
blisibimod Immunopharmacology Ligand 9518 A-623, AGP3 peptibody, AMG 623, Fc-Agp-3
BOC-ATE 2042
BODIPY® TMR-NMU 3858
bombesin 616
[Bpa1,Ile13]motilin (human) 1452
[Bpa6,Tyr10]secretin-27 (rat) Ligand is labelled Ligand is radioactive 1154
BP-CCL3 752 BP-LD78α, BP-MIP-1α, photoactivatable macrophage inflammatory protein-1α
BPTI-K15R/R17G 7897
BQ123 997 BQ 123, BQ-123
BQ 3020 3859 BQ-3020, BQ3020
[125I]BQ3020 Ligand is labelled Ligand is radioactive 1005 [125I]-BQ3020
[3H]BQ123 Ligand is labelled Ligand is radioactive 1003 [3H]-BQ123, [3H]cyc(DTrp-DAsp-Pro-DVal-Leu
bremelanotide Approved drug 10408 PT-141, PT141, Vyleesi®
brimapitide Immunopharmacology Ligand 9101 AM-111, D-JNKI-1, XG-102
B-R13/17K H2 relaxin 4371 AT-001, B13/17K H2 relaxin
α-bungarotoxin 3964
[125I]α-bungarotoxin Ligand is labelled Ligand is radioactive 3972
[3H]α-bungarotoxin Ligand is labelled Ligand is radioactive 3981
buserelin Approved drug 3860 buserelin acetate, HOE 766, HOE 766A, ICI 123215, Metrelef®, Suprefact®
[125I]buserelin Ligand is labelled Ligand is radioactive 1167 [125I]-buserelin
Bv8 5362 Bombina variegata protein
[Bz-Phe6]U-II (human) 2159 human [Bz-Phe6] urotensin-II
 
C Back to top
C089 5779
C21 7037
C3 1291
C7 3861 galanin(1-13)spantide
C5a hexapeptide analogue 5768 Phe-Lys-Ala-dCha-Cha-dArg
[125I]C3a (human) Ligand is labelled Ligand is radioactive 3773 [125I]-C3a
[125I]C5a (human) Ligand is labelled Ligand is radioactive 3774 [125I]-C5a
calciseptine 4149
calcitonin (salmon) Approved drug 6973 CT (salmon), Miacalcin®
cANF4-23 4892 des[Gln18,Ser19,Gly20,Leu21,Gly22]ANP4οΎ–23-NH2
cangitoxin II 7568 cangitoxin-2, cangitoxin-II, CGTX-II
C5apep 11344
carbetocin Approved drug 11169 Pabal®
CARTPT (76-96) 10571
casoxin C 10224
[125I]cathepsin G (human) Ligand is labelled Ligand is radioactive 1017 [125I]cathepsin G
CB-182804 11003 CB-182,804, CB182804
CCK-58  {Sp: Dog} 862
[3H]CCK-8 (human, mouse, rat) Ligand is labelled Ligand is radioactive 4765 [3H]-CCK-8
[125I]CCL11 (human) Ligand is labelled Ligand is radioactive 794 [125I]eotaxin
[125I]CCL16 (human) Ligand is labelled Ligand is radioactive 1275 [125I]LEC
[125I]CCL17 (human) Ligand is labelled Ligand is radioactive 3652 [125I]TARC
[125I]CCL19 (human) Ligand is labelled Ligand is radioactive 3655 [125I]ELC
[125I]CCL1 (human) Ligand is labelled Ligand is radioactive 814 [125I]I-309, [125I]P500, [125I]TCA-3
[125I]CCL20 (human) Ligand is labelled Ligand is radioactive 3654 [125I]LARC, [125I]MIP-3α
[125I]CCL21 (human) Ligand is labelled Ligand is radioactive 3656 [125I]SLC
[125I]CCL25 (human) Ligand is labelled Ligand is radioactive 3657 [125I]TECK
[125I]CCL27 (human) Ligand is labelled Ligand is radioactive 3653 [125I]CTACK
[125I]CCL2 (human) Ligand is labelled Ligand is radioactive 762 [125I]MCAF, [125I]MCP-1, [125I]monocyte chemotactic protein-1
[125I]CCL3 (human) Ligand is labelled Ligand is radioactive 763 [125I]macrophage inflammatory protein-1α, [125I]MIP-1α
[125I]CCL4 (human) Ligand is labelled Ligand is radioactive 799 [125I]macrophage inflammatory protein-1β, [125I]MIP-1β
[125I]CCL5 (human) Ligand is labelled Ligand is radioactive 764 [125I]RANTES, [125I]regulated upon activation normal T cell expressed and secreted
[125I]CCL7 (human) Ligand is labelled Ligand is radioactive 765 [125I]MCP-3, [125I]monocyte chemotactic protein-3
[125I]CCL8 (human) Ligand is labelled Ligand is radioactive 766 [125I]MCP-2, [125I]monocyte chemotactic protein-2
[125I]CCL1 (mouse) Ligand is labelled Ligand is radioactive 5546
CCL20-SEAP(His)6 809 LARC fused with secreted alkaline phosphatase, LARC-SEAP(His)6, MIP-3α fused with secreted alkaline phosphatase
cenderitide 9066 CD-NP
cetrorelix Approved drug Immunopharmacology Ligand 1190 Cetrotide®, SB-075
[125I]cetrorelix Ligand is labelled Ligand is radioactive 1186
CGEN-856 7041 P61
CGEN-857 7040 P33
CGEN-855A 6241
CGP 23996 2005 CGP-23996, CGP23996
CGP42112 3944 CGP 42112, CGP 42112A
[125I]CGP 23996 Ligand is labelled Ligand is radioactive 2022
[125I]CGP42112 Ligand is labelled Ligand is radioactive 594 [125I]-CGP42112, Cgp 42112B, Cgp-42112A
α-CGRP-(8-37) (human) 700 α-CGRP (8-37) (human), human α-calcitonin gene-related peptide (8-37)
[125I]αCGRP (human) Ligand is labelled Ligand is radioactive 3766 [125I]-αcalcitonin gene-related peptide, [125I]-αCGRP
[125I]αCGRP (mouse, rat) Ligand is labelled Ligand is radioactive 6567
α-CGRP-(8-37) (rat) 701 α-CGRP (8-37) (rat), rat α-calcitonin gene-related peptide (8-37)
CH 275 2006 CH-275, desAA1,2,5[D-Trp8,IAmp9]somatostatin-14
charybdotoxin 2328 ChTX
charybdotoxin-GLU32 analog 2329 ChTX-GLU32
[Cha6]U-II-(4-11) 9439
chemerin C-terminal peptide 3422 bioactive chemerin peptide, chemerin 149-157, chemerin 9, chemerin-9
CHIPS 3724 chemotaxis inhibitory protein of S. aureus
CHIPS-(28-149) 5770 CHIPS28-149
[125I]CHIPS Ligand is labelled Ligand is radioactive 1027 [125I]chemotaxis inhibitory protein of S. aureus
[(CH2NH)4,5]secretin 3755 [ψ4,5]secretin
[125I]chorionic gonadotropin (human) Ligand is labelled Ligand is radioactive 3775 [125I]CG (human), [125I]-CG, [125I]-chorionic gonadotropin
cibinetide Immunopharmacology Ligand 9677 ARA 290, ARA-290, PH-BSP, PHBSP
C12-iE-DAP 9508
cilengitide 6597 EMD-12192, EMD-121974
4-Cl-cinnamoyl-c[DCys-4Pal-DTrp-Orn-Val-Cys]-His-amide 2161
[125I]CNP (human) Ligand is labelled Ligand is radioactive 4847 [125I]-CNP
C2-NPY (pig) 1534
compound 6b [PMID: 24999562] 7927
compound 3c [PMID: 30360354] Immunopharmacology Ligand 10591 [As(4-F)F4]-GHRP-6, azasulfuryl-p-fluorophenylalanine-4-[As(4-F)F4]-GHRP-6, H-His-D-Trp-Ala-(4-F)AsF-D-Phe-Lys-NH2
compound 5d [PMID: 25815150] 9008
compound 8d [PMID: 24999562] 7926
compound 1 [PMID: 25241924] 7801
compound 2 [PMID: 11375253]