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The IUPHAR/BPS Guide to PHARMACOLOGY complete ligand list

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Antibacterial ligands
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Ligand name ID Synonyms
A Back to top
A2315A 10846
acorafloxacin 10753 avarofloxacin (former name), JNJ-Q2, JNJQ2
afabicin 10754 AFN-1720, Debio 1450, Debio1450
AHPN 3431 CD 437, CD437, Ro 47-2077
alafosfalin PDB Ligand 9503 alaphosphin
alalevonadifloxacin 10756 WCK 2349, WCK-2349, WCK2349
alpibectir 12957 BVL-GSK098
Altromycin B 10964
amifloxacin 10758 compound 7 [PMID: 2834557], WIN 49, 375, WIN 49,375-3, WIN-49375, WIN49375
amikacin Approved drug PDB Ligand 10894 Amikin®, AMK, Arikayce liposomal®, BB-K8
amoxicillin Approved drug 10895 Amoxil®, BRL-2333, co-amoxiclav (amoxicillin + clavulanic acid), Moxatag®, NSC-277174, Trimox®
ampicillin Approved drug PDB Ligand 10896 aminobenzylpenicillin, KS-R1, Penbritin®, Polycillin, Principen®
AN0128 10983 AN 0128, AN-0128, compound 2g [PMID: 16997550]
ancremonam 13161 BOS-228, LYS228
ANT3310 12795
apalcillin 10759 PC-904, PC904, WY-44,417, WY-44417
apramycin PDB Ligand 10760 EBL-1003, EL-857, EL857, nebramycin factor 2, nebramycin II
arachidonic acid PDB Ligand 2391 C20:4
arbekacin Approved drug PDB Ligand 7345 arbekacin sulfate, habekacin, ME1100, NPC-14
aspoxicillin Approved drug 12293 Doyle®, TA-058
avibactam Approved drug PDB Ligand 10761 AVI, NXL 104, NXL-104, NXL104
avibactam tomilopil 12949 ARX-1796, AV-006, PF-07338233
azidamfenicol Approved drug 12397 azidamphenicol, azidoamfenicol, azidoamphenicol, Thilocof®
azidocillin 12291 BRL 2534, SPC 297 D
azithromycin Approved drug PDB Ligand Immunopharmacology Ligand Antimalarial Ligand 6510
azlocillin Approved drug 12260 Azlin®, BAY-E-6905
aztreonam Approved drug 10763 Azactam®, Cayston®, SQ 26776, SQ-26776, SQ26776
 
B Back to top
bacampicillin Approved drug 12292 Penglobe®, Spectrobid®
bacitracin A Approved drug 12812
BAL19403 10981 BAL 19403, BAL-19403
BAL30072 11004 BAL-30072
balofloxacin Approved drug 13105 Q-35, Q-Roxin®
BAS-118 10976 BAS118, compound 7n [PMID: 11728192]
BB2-50F PDB Ligand 13072
BC-3205 10998
BC-7013 11034 BC7013
bedaquiline Approved drug PDB Ligand 11171 BDQ, compound 1a [PMID: 17496888], R-207910, Sirturo®, TMC-207, TMC207
bederocin PDB Ligand 10764 REP-8839, REP8839
bekanamycin Approved drug PDB Ligand 12182 kanamycin B, nebramycin V
benapenem 12793
besifloxacin Approved drug 12877 Besivance®, BOL-303224-A, ISV-403, SS734
beta-defensin 4A 3648 beta-defensin 2, HBD2, skin-antimicrobial peptide 1 (SAP1)
biapenem Approved drug 12022 L-627, LJC10,627, Omegacin®, RPX2003
BLI-489 free acid 10995 BLI489
bluensomycin 10765 bluensin, U-12898, U12898
borrelidin Antimalarial Ligand 11306 (-)-borrelidin
BRL-42715 10993 C6-(N1-Methyl-1,2,3-trazolylmethylene)penem, LS-186900 (sodium salt), LS-187554
BRL-44154 11036 analogue 4f [Brown et al., 1991], BRL44154
brodimoprim 12325 Ro 10-5970
BTZ-043 13034 BTZ-10526043, MMV676603
butikacin 10766 UK-18,892, UK-18892, UK18892
BWC0977 12809
 
C Back to top
cadazolid PDB Ligand 10767 ACT-179811, ACT179811
caffeic acid PDB Ligand 5155
capreomycin IB Approved drug 13256 Capastat®
carbenicillin Approved drug 10768 BRL-2064, BRL2064, carboxybenzylpenicillin, CBPC, CP 15639-2, CP-156392, Pyopen®
carfecillin Approved drug 12288 BRL 3475, carbenicillin phenyl, Uticillin®
carindacillin Approved drug 12276 carbenicillin indanyl, CP-15,464-2, CP-15464-2, Geocillin®
carumonam Approved drug 12296 AMA-1080, Ro 17-2301
cationomycin 11002 BRN-6263205, BRN6263205, LS-52659, LS52659
CB-182804 11003 CB-182,804, CB182804
cefacetrile 12192 Celospor®, cephacetrile
cefaclor Approved drug 10897 Ceclor®, Lilly 99638, Raniclor®
cefadroxil Approved drug 4831 Duricef®
cefaloglycin Approved drug 12193 cephaloglycin, Kafocin®
cefaloridine 12189 cephaloridine, ceporin
cefalotin Approved drug PDB Ligand 8798 cephalothin, cephalotin, Keflin®
cefamandole Approved drug PDB Ligand 12210 cephamandole
cefapirin Approved drug 12191 Cefadyl®, cephapirin
cefatrizine 12204 BL-S640
cefazaflur 10770 SK&F 59962
cefazedone 12203 EMD-30087, Refosporen®
cefazolin 10935 Ancef®, cephazolin, CEZ, Kefzol®, SK&F-41558
cefbuperazone 12253
cefcapene Approved drug 12053 Flomox® (cefcapene pivoxil), S-1006
cefclidin 10771 cefclidine, E-1040, E1040
cefdinir Approved drug 12023 FK 482, Omnicef®
cefditoren Approved drug 12030 ME 1206, Spectracef® (cefditoren pivoxil)
cefepime Approved drug 10772 BMY-28142, BMY28142, CFPM, Maxipime®, Renapime®
cefetamet 12416 Ro 15-8074
cefetecol 10775 GR-69153, GR-69153X, GR69153
cefiderocol Approved drug 10776 compound 3 [PMID: 29960205], Fetcroja®, Fetroja®, GSK-2696266, GSK2696266, RSC 649266, RSC-649266, RSC649266, S-649266
cefixime Approved drug PDB Ligand 10898 (E)-Cefixime, Cefspan®, CFIX, FK-027, FR-17027, Suprax®
cefluprenam 10777 E-1077, E1077
cefmatilen 10778 S-1090, S1090
cefmenoxime Approved drug 12024 A-50912, Abbott 50192, Bestron®, Cefmax®, SCE-1365
cefmetazole Approved drug PDB Ligand 12215 CS-1170, U-72791, Zefazone®
cefminox 12255 MT 141
cefodizime 12032 HR 221
cefonicid Approved drug 12217 Monocid®, SK&F 75073
cefoperazone Approved drug 12025 Cefobid®, T-1551
ceforanide Approved drug 12218 BL-S786, Precef®
cefoselis Approved drug 12034 FK-037, Wincef®
cefotaxime Approved drug PDB Ligand 10893 Claforan®, Ru-24756
cefotetan Approved drug 10936 Apatef®, Cefotan®, ICI-156834, ICI156834
cefotiam 12254 SCE 963
cefoxitin Approved drug PDB Ligand 10937 Cenomycin®, CFX, Mefoxin®, MK-306, MK306
cefozopran Approved drug 12054 SCE-2787
cefpimizole 10779 CPIZ, U 63196E, U-63,196, U-63196E
cefpiramide Approved drug 12027 SM-1652, WY-44635
cefpirome Approved drug 12033 HR 810, Romecef®
cefpodoxime Approved drug 10780 RU-51746, Vantin®
cefprozil Approved drug 12219 BMY-28100, Cefzil®
cefsulodin 10783 Cefonomil®, CGP-7174-E, CGP7174/E
ceftaroline fosamil Approved drug 10899 PPI-0903, TAK-599, Teflaro®, Zinforo®
ceftazidime Approved drug 10762 CAZ, Fortaz®, Fortum®, GR 20263, GR-20263, GR20263, LY-139381, LY139381, Pentacef®, Tazicef®
cefteram Approved drug 11051 cefterame, ceftetrame, CFTM, Ro 19-5247, T-2525
ceftezole 12259 ceftezol, FR10123
ceftibuten Approved drug 12029 7432-S, Cedax®, SCH 39720
ceftiolene 10784 42980RP, cefatiolene, RP 42,980, RP 42980, RP-42980, RP42980
ceftizoxime Approved drug 10785 Cefizox®, compound 22 {PMID: 2342058], Epocelin®, FK-749, FK749, FR-13749, FR13749, SK&F 88373-Z
ceftizoxime alapivoxil 10786 AS-924, AS924, KY-020, KY020
ceftobiprole Approved drug 10787 BAL-9141, BAL9141, BAL9141-000, BAL9141000, Ro-63-9141, Ro-639141, Zeftera®, Zevtera®
ceftolozane Approved drug 10788 CXA-101, CXA101, FR-264205, FR264205, Zerbaxa® (ceftolozane + tazobactam)
ceftriaxone Approved drug 5326 Rocephin®
cefuroxime Approved drug PDB Ligand 10900 Ceftin®, CXM, Kefurox®, Zinacef®
cephalexin Approved drug 4832 cefalexin, Ceporex®, Keflex®
cephalosporin P1 12330 acremonic acid
cephradine Approved drug 4830 cefradine, Infexin®, Velocef®
cetefloxacin 10790 compound 43f [PMID: 7990118], E-4868, E4868
cethromycin PDB Ligand 10791 A-195773, Abbott-195773, ABT-773, ABT773, Restanza®
cetocycline 10792 A-40728, Abbott 40728, chelocardin, compound 1 [PMID: 379332]
CG-400549 PDB Ligand 10984 CG400549
CGP-31608 10963 CGP 31608, CGP31608
chalcomycin 11058
chinfloxacin 11017
chloramphenicol Approved drug PDB Ligand 10901 Brolene®, chloromycetin
chlorocardicin 11044
chrysin PDB Ligand 8789 NSC-407436
cilastatin Approved drug 5166 MK 0791, MK-791, MK791, Primaxin®
cinoxacin Approved drug 12401 Cinobac®, Lilly 64716
ciprofloxacin Approved drug PDB Ligand 10902 BAY-O-9867, BAY-O9867, Cetraxal®, Ciloxan®, Cipro®, CPFX, Proquin XR
CJ-15,801 Antimalarial Ligand 10610 CJ-15801
cladosporin PDB Ligand Antimalarial Ligand 10247 asperentin
clarithromycin Approved drug PDB Ligand 10903 6-O-methylerythromycin, A-56268, ABBOTT-56268, Biaxin®, Klaricid®, TE-031
clavulanic acid Approved drug PDB Ligand 11128 BRL-14151, BRL-14151K, BRL14151, clavulanate, MM 14151
clinafloxacin 10793 AM 1091, CI-960, PD-127321
clindamycin Approved drug PDB Ligand Antimalarial Ligand 10607
clofazimine Approved drug Immunopharmacology Ligand 9184 Lamprene®
clofoctol Approved drug 12926 Gramplus®, Octofene®
clometocillin 12294 clometacillin, clomethacillin
clorobiocin PDB Ligand 12127 chlorobiocin, RP 18,631
clovibactin 13080 Novo29
cloxacillin Approved drug PDB Ligand 11126 BRL-1621, BRL1621, chloroxacillin, Methocillin S, Syntarpen®, Tegopen®
colistin Approved drug 10794 Colobreathe®, polymyxin E, Promixin®
compound 16 [PMID: 38385364] 13259
compound 5 [Stecula et al., 2020] 11155 MCULE-2879769428
contezolid Approved drug PDB Ligand 10795 MRX-1, MRX-I, Youxitai®
contezolid acefosamil (parent) 10796 MRX-4
Corallopyronin A 11029 CorA, LS-54950, LS54950
coumamycin PDB Ligand 10879 coumermycin A1, notomycin
CRS3123 PDB Ligand 10991 CRS-3123, REP-3123, REP3123
cyclacillin Approved drug 4817 ciclacillin, Cyclapen®, Vastcillin®, Wy-4508
cyclothialidine 10988 Ro 09-1437
 
D Back to top
dactimicin 11001 Formimidoyl-fortimicin A, SF-2052, SF2052
dalbavancin Approved drug 10876 BI-397, BI397, Dalvance®, Xydalba®
dalfopristin Approved drug PDB Ligand 10797 RP-54476, RP54476, Synercid® (dalfopristin + quinupristin)
danirixin Immunopharmacology Ligand 8500 GSK-1325756B, GSK1325756, GSK1325756B
dapsone Approved drug Antimalarial Ligand 10934 Aczone®, NSC-6091
daptomycin Approved drug 10904 Cubicin®, LY-146032, LY146032
DC-159a 10982
D-cycloserine Approved drug PDB Ligand 9489 Seromycin®
DEBIO 1452 10755 afabicin desphosphono, AFN-1252, AFN-12520000, DEBIO-1452, DEBIO1452
decaplanin 10968 M 861410, M86-1410, MM-47761
declovanillobiocin 12128 novclobiocin 313
delafloxacin Approved drug PDB Ligand 10799 Abbott 492, ABT-492, ABT492, Baxdela®, Quofenix®
delamanid Approved drug 12876 Deltyba®, OPC-67683
delpazolid 10999 LCB-01,0371, LCB-01-0371, LCB01-0371
demeclocycline 10905 Declomycin®, Ledermycin®
diacerein Approved drug 10800 Artrodar®, Fisiodar®
dibekacin Approved drug PDB Ligand 12134 3',4'-dideoxykanamycin B, debecacin
dicloxacillin Approved drug 12261 BRL-1702, Diclocil®, Dynapen®
difficidin 11062
difloxacin 10801 A 56619, A-56619, Dicural®
dihydrostreptomycin Approved drug PDB Ligand 12163
dihydroxybenzofuran 10992 2,3-Benzofurandiol
dirithromycin Approved drug PDB Ligand 12928 AS-E 136, Dynabac®, LY237216
DK-507k 11037
doripenem Approved drug PDB Ligand 12183 compound 1m [PMID: 8621362], Doribax®, S-4661
doxycycline Approved drug PDB Ligand Immunopharmacology Ligand Antimalarial Ligand 6464 BMY-28689, Monodox®, Vibramycin®
DS-8587 10955 DS8587
DS-2969b 10985 DS 11960558 (DS-2969b prodrug), DS-2969, example 2 [WO2017/056012A1]
Dup-105 10950 DuP 105, DuP105
DuP-721 10960 DuP 721
durlobactam Approved drug 12693 ETX-2514, EXT2514, Xacduro® (sulbactam and durlobactam)
DX-619 11039 compound 4 [PMID: 19736016], DX619
 
E Back to top
E-0702 11056
ecenofloxacin 10802 CFC-222, CFC222
E-1010 free base 11050 E1010, ER-35786
Enduracidin 10989
enmetazobactam Approved drug 12188 AAI101, OCID-5090
enoxacin Approved drug 8882 AT-2266, CI-919, Penetrex®
enteromycin carboxamide 11063 BRN 2416858, BRN-2416858, BRN2416858, LS-14645
enviomycin Approved drug 13276 Tuberactin®, tuberactinomycin N
eperezolid 10803 comound 2 [PMID: 23584544], PNU-100592, PNU100592, U-100592, U100592
epetraborole 13079 AN3365, GSK2251052
epicillin 10804 Dexacillin®, SQ 11302, SQ-11302, SQ11302
epiroprim 12327 Ro 11-8958, TCMDC-137295
eravacycline Approved drug PDB Ligand 10805 compound 17j [PMID: 2148514], TP-434, TP434, Xerava®
eremomycin 10959 A82846A
ertapenem Approved drug 10906 Invanz®, L-749345, MK-0826, MK-826
erythromycin Approved drug PDB Ligand 1456 EM-A, E-Mycin®, Erythrocin®, erythromycin-A
ethambutol Approved drug PDB Ligand 12996 Myambutol®
etheromycin 10994 CP‐38 295
ethionamide Approved drug PDB Ligand 12954 1314 TH, Bayer 5312, Trecator®
ethyl bromopyruvate 10952
ETX0282 10781 ETX-0282
ETX0462 PDB Ligand 11753 ETX-0462, VMM
ETX1317 10782 ETX-1317
evernimicin 10806 SCH 27899, SCH-27899, SCH27899, Ziracin®
evybactin 12922 GLXC-26146
 
F Back to top
fandofloxacin 10807 DW-116, DW116
faropenem PDB Ligand 10808 compound 1 [PMID: 9216830], faropenem medoxomil, fropenem
feldamycin 10979 BMY-28565, BMY28565, U-48266
Ferrimycin A1 10966
ficellomycin 10965 U-47,929, U-47929, U47929
fidaxomicin Approved drug PDB Ligand 10909 Dificid®, Dificlir®, lipiarmycin, OPT-80, PAR-101, tiacumicin B
finafloxacin 10809 AL-60371, AL60371, Xtoro®
fleroxacin Approved drug 12476 AM-833, Megalone®, Quinodis®, Ro 23-6240
flomoxef 12251 6315-S, Flumarin®
florfenicol 12923 SCH 25298
flucloxacillin Approved drug 10910 BRL-2039, BRL2039, floxacillin
fludalanine 10810 3-fluoro-D-alanine, MK-0642, MK0642
flurithromycin Approved drug 12927 (8S)-8-fluoroerythromycin A, P-0501A
fobrepodacin 13062 pVXc-486, SPR720
fosfomycin Approved drug PDB Ligand 10813 Monurol®, phosphomycin, phosphonomycin, Veramina®
fosmidomycin PDB Ligand Antimalarial Ligand 9739 FR-31564
funobactam 13114 XNW4107
furagin Approved drug 12367 furazidin, furazidine, NF416
furazolidone Approved drug 12343 Furoxone®
furazolium 10814 Novofur
fusidic acid Approved drug PDB Ligand 10815 CEM-102, CEM102, Fucidin®, fusidate, sodium fusidate, Taksta®
 
G Back to top
ganfeborole 12796 GSK3036656, GSK656
garenoxacin Approved drug 12402 BMS-284756, Ganefloxacin, Garenfloxacin, Geninax®, T-3811
gatifloxacin Approved drug 10816 AM-1155, AM1155, Gatiflo®, GTFX, Tequin®, Zymar®
gemifloxacin Approved drug 12406 Factive®, LB20304, SB 265805
gentamicin Approved drug 2427 Garamycin®, gentamicin sulfate
gepotidacin PDB Ligand 10817 GSK-2140944, GSK2140944
gloximonam 10880 SQ 82,531
grepafloxacin Approved drug 10818 OPC 17116, OPC-17116, OPC17116, Raxar®
GSK2556286 13078 GSK286
GT-1 13251 LCB10-0200
 
H Back to top
hedamycin 10958 antibiotic B 26,158, B26158, NSC-70929
helvolic acid 12329 fumigacin
hesperetin PDB Ligand 10953 3',5,7-Trihydroxy-4'-methoxyflavanone, NP-13, NSC-57654
hetacillin Approved drug 12263
hexachlorophene Approved drug PDB Ligand 11069 Inh 1 [PMID: 32284327], Nabac®
HSGN-218 13054
ω-Hydroxyemodin 11005 Citreorosein, omega-Hydroxyemodin
hymeglusin 5886 antibiotic 1233A, F-244, L-659,699
 
I Back to top
ibafloxacin 10819 R-835, R835, S-25930, S25930
ibezapolstat 11030 ACX-362E, ACX362E
iboxamycin 11790 IBX, OPP-3
iclaprim 10820 AR-100, AR100, Mersarex®, RO-48-2622, RO-482622
imipenem Approved drug 10821 MK-0787, MK0787, Primaxin® (imipenem + cilastatin), Recarbrio® (imipenem + cilastatin + relebactam).
indanomycin 10949 X-14547A
indolmycin PDB Ligand Antimalarial Ligand 11021 PA 155 A, PA-155-A, PA-155A, TAK-083
Irresistin-16 10973 IRS-16, IRS16
iseganan 10822 IB-367, IB-367-03
isepamicin Approved drug 12136 HAPA-B, Sch 21420
isoniazid Approved drug PDB Ligand 12761 isonicotinic acid hydrazide, Nydrazid®, Rimifon®
isovanillobiocin 12129 novclobiocin 312
IT-62-B 11032
ivermectin Approved drug 2373 Heartgard®, ivermectin B1a, MK-933, Sklice®, Soolantra®
 
J Back to top
josamycin Approved drug 12924 kitasamycin A3, leucomycin A3, turimycin A5
 
K Back to top
kaempferol PDB Ligand 11052 Robigenin
kanamycin Approved drug PDB Ligand 12132 kanamycin A
Katanosin B 10970 Lysobactin
KB-5246 11046 KB5246, LS-99630
kibdelomycin A 11016
 
L Back to top
L-701677 11042 L-701,677
L-708365 10980 L 708,365, L 708365, L-708,365
lactivicin 11022 compound 1 [PMID: 17676039], LTV
lascufloxacin 10823 KRP-AM1977
latamoxef Approved drug 12031 6059-S, LY127935, moxalactam, Moxam®
LBM-415 11043 LBM415, NVP LBM-415, NVP-PDF-713, PDF-713, VIC-104959
L-cycloserine Approved drug 9488 levcycloserine, Seromycin®
ledaborbactam 13082 VNRX-5236
lefamulin Approved drug PDB Ligand 10824 BC-3781, BC3781, compound 7 [PMID: 24874438], Xenleta®
leinamycin 11041 DC-107, DC107
lenapenem 10825 BO-2727, BO2727, L-739,428, L-739428
levofloxacin Approved drug PDB Ligand 10911 DR-3355, Levaquin®, Quinsair®
levonadifloxacin 10757 (S)-(-)-nadifloxacin, WCK 771, WCK-771, WCK771
levopropicillin 10826 BRL-284, BRL284, L-Propicillin, P-248, P248
lincomycin Approved drug PDB Ligand 10941 Bactramycin®, L-Mycin®, LCM, Lincocin®, Lincorex®, U 10,149A, U-10149
linezolid Approved drug PDB Ligand 10827 PNU-100766, PNU100766, U-100,766, U-100766, ZLD, Zyvox®
lomefloxacin Approved drug 12407 Maxaquin®, NY-198, SC-47111, Uniquin®
loracarbef Approved drug 12247 KT-3777, Lorabid®, LY163892
luminamicin 11053 coloradocin, LS-90907
lymecycline Approved drug 10912 N-Lysinomethyltetracycline, tetracycline-L Methylene-Lysine, Tetralysal®
lysinomicin 10969
 
M Back to top
M14659 11047 GR 63116, GR-63116, M 14659, M-14659
macozinone 13055 PBTZ169
Macquarimicin A 10978
mafenide Approved drug PDB Ligand 12697 homosulfanilamide, Sulfamylon®
maridomycin 10828 LS-87912, Maridomycin III
MC-02479 11033 MC 02479, MC02479, RWJ 54428, RWJ-54428
ME-1228 acid 11045 ME1228
mecillinam Approved drug 12813 amdinocillin, Coactin®, FL 1060, Selexidin®
meropenem Approved drug PDB Ligand 10829 ICI 194,660, Merrem®, SM-7338
mersacidin 11014 M87 1551, M87-1551
metampicillin 12274 methampicillin, methylenampicillin, Micinovo®, Viderpen®
methenamine Approved drug 10913 Hiprex®, Mandelamine®, Urex®
methicillin Approved drug PDB Ligand 12264 meticillin
metronidazole Approved drug PDB Ligand 10914 BAY-5360, BAYER 5360, Flagyl®, Metrogel®, ROZEX®
mezlocillin Approved drug 12272 BAYPEN®, Mezlin®, Multocillin®
MGB-BP-3 10996 compound 50 [PMID: 17960927], MGB-BP3
micronomicin Approved drug 12162 gentamicin C2b, Sagamicin®, XK-62-2
midecamycin Approved drug 13158 espinomycin A, platenomycin B1, rubimycin, SF-837, turimycin P3
mideplanin 10830 CTA A1, MDL 62873, MDL-62873, MDL62873
minocycline Approved drug 10831 CL 59806, CL-59806, CL59806, Dynacin®, MINO, Minocin®, NSC-141993
modithromycin 13000 EDP-420, EP-013420, S-013420
moxifloxacin Approved drug PDB Ligand 10915 Avelox®, BAY-12-8039, BAY-128039, BAY128039, MFX, MOXIVIG® (opthalmic solution)
mupirocin Approved drug PDB Ligand Antimalarial Ligand 10916 Bactroban®, BRL-4910A, BRL-4910F, Centany®, pseudomonic acid
murepavadin 10832 POL7080, RG-7929, RG7929, RO-7033877, RO7033877
MUT056399 PDB Ligand 11000 Fab-001, FAB001, MUT-056399
 
N Back to top
nacubactam 10833 OP-0595, OP0595, RG-6080, RG6080, RO-7079901, RO7079901
nadifloxacin Approved drug 12919 Nadixa®, OPC-7251
nafcillin Approved drug 10942 Ethoxynaphthamido Penicillin Sodium, Nallpen®, Unipen®
nafithromycin 10834 WCK 4873, WCK-4873, WCK4873
nalidixic acid Approved drug PDB Ligand 12773 NegGram®, Win 18,320
napsamycin C 11008
napsamycin D 11009
narasin 10835 C-7819B, Lilly 79891, Monteban®, Narasin A
nemonoxacin Approved drug 10836 Taigexyn®, TG-873870, TG873870
neomycin Approved drug PDB Ligand 709 Neo-Rx®, neomycin sulfate
neopyrrolomycin 10962
netilmicin Approved drug 12159 1-N-ethylsisomicin, Sch 20569
niclosamide Approved drug PDB Ligand 8494 VU0243604
nifuratel Approved drug 12348 Macmiror®, Magmilor®, methylmercadone
nifuroxazide Approved drug 12358 NSC-759261, RC-27109, SJ000287313
nifurprazine 10837 carofur, HB-115, HB115
nifurquinazol 12344 NF-1088
nifurtimox Approved drug 12364 BAY 2502, BAY A2502, Bayer 2502, Lampit®
nifurtoinol Approved drug 12346 hydroxymethylnitrofurantoin, Urfadyn PL®
nifurzide 12365 Ricridene®
nitrofural Approved drug PDB Ligand 12366 Furacin®, Furacine®, nitrofurazone
nitrofurantoin Approved drug PDB Ligand 10917 Furadantin®, Macrobid®, Macrodantin®, Nitro Macro®, NSC-2107, NSC-44150
nocardicin A 12295
nodusmicin 11019 nodusmicin 1
nojirimycin 10951 5-amino-5-deoxy-D-glucopyranose, D-gluco-piperidinose
norfloxacin Approved drug 12408 AM-715, Chibroxin®, MK-0366, Noroxin®
NOSO-502 13157
novclobiocin 101 12131
novobiocin Approved drug PDB Ligand 12021 Albamycin®, cardelmycin, cathomycin, PA 93, streptonivicin
NPS 2143 PDB Ligand 716 NPS-2143, NPS2143
NSC-84963 10956 NSC 84963, NSC84963
NSC-93169 10957 NSC 93169, NSC93169
 
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ofloxacin Approved drug 10918 DL-8280, Exocin® (eye drops), Floxin®, HOE-280, OFX, Tarivid®
olamufloxacin 10838 HSR-903, HSR903
oleandomycin Approved drug 13280 amimycin, landomycin, Matromycin®, P.A.105, Romicil®
oleuropein 11027
olivanic acid 12811
omadacycline Approved drug PDB Ligand 10839 amadacycline, compound 6 [PMID: 21302930], Nuzyra®, PTK-0796, PTK0796
OPS-2071 13197
oritavancin Approved drug 10877 Kimyrsa®, LY-333328, LY333328, Orbactiv®
oxacillin Approved drug 10943 Bactocill®
oxantel Approved drug 10840 CP-14,445, CP-14445
oxaquin 10997 DNV-3837, DNV3837, MCB-3837, MCB3837
oximonam 12297 SQ 82,291
oxolinic acid Approved drug PDB Ligand 12999
oxytetracycline Approved drug PDB Ligand 10919 E703, NSC-9169, Terramycin®
ozenoxacin Approved drug 10841 Ozadub®, T-3912, T3912, Xepi®
 
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pafuramidine 10842 DB-289, DB289
paldimycin 10843 Antibiotic 273 A, U-70,138, U-70138F
panipenem Approved drug 12184 Carbenin® (panipenem + betamipron), CS-533, RS-533
paromomycin Approved drug PDB Ligand 12160 aminosidine, catenulin, Humatin®, monomycin A
pazufloxacin Approved drug 12410 Pasil®, Pazucross®, T-3761
pefloxacin Approved drug 12411 1589 RB, AM-725
penamecillin Approved drug 12808 Havapen®, WY-20788
penicillin G Approved drug PDB Ligand 4796 penicillin G sodium, penicillin-G potassium
pheneticillin Approved drug 12275 alfacilin, Broxil®, feneticillin, phenethicillin
phenoxymethylpenicillin Approved drug PDB Ligand 10920 Oracillin®, PC Pen VK®, Pen-V®, penicillin V, Penicillin VK, PNV
phleomycin 10954 NSC 61586, NSC-61586
pipemidic acid Approved drug 12774 Pipram®
piperacillin Approved drug PDB Ligand 10921 CL 227,193, CL-227193, PIPC, T-1220, Tazocin® (piperacillin + tazobactam)
pirazmonam 10844 compound 2 [PMID: 25658376], SQ 83,360, SQ-83360, SQ83360
pirbenicillin 10845 CP-33,994, CP-33,994-2
piromidic acid Approved drug 12475 Bactramyl®, Panacid®, PD-93
pivampicillin 12920 MK-191, Pondocillin®
pivmecillinam Approved drug 10922 amdinocillin pivoxil, pivmecillinam hydrochloride, RO-10-9071, RO-109071, Selexid®
plazomicin Approved drug PDB Ligand 10847 ACHN-490, ACHN490, Zemdri®
pleuromulin 12935 drosophilin B, pleuromutilin
plusbacin A3 11020
PNU-288034 10977 compound 2 [PMID: 16644216], PNU288034
polymyxin B Approved drug 10338 Aerosporin®
posizolid 12762 AZD2563, AZD5847
poststatin 10967 L-Val-L-Val-3-amino-2-oxo-valeryl-D-Leu-L-Val
pralurbactam 13037
premafloxacin 10848 compound 21 [PMID: 17303420], U-95376, U95376
pretomanid Approved drug 11172 PA-824, PA824
pristinamycin IA Approved drug 12934 mikamycin B, ostreogrycin B, Pyostacine®, streptogramin B, virginiamycin B
pristinamycin IIA Approved drug PDB Ligand 12933 mikamycin A, ostreogrycin A, Pyostacine®, streptogramin A, virginiamycin M1
prontosil 12743 prontosil red, prontosil rubrum, sulfamidochrysoidine
prulifloxacin Approved drug 12860 NM441
pyrazinamide Approved drug PDB Ligand 7287 aldinamide, Zinamide®
 
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QPX7831 13241
quabodepistat 13059 OPC-167832
quinupristin Approved drug 10798 RP 57669, RP-57669, RP57669, Synercid® (dalfopristin + quinupristin)
 
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radezolid PDB Ligand 10849 Rx-01_667, RX-103, RX-1741, RX103, RX1741
ranbezolid 11007 RBx 7644
rancinamycin IA 11015 Rancomycin 1, U-22583, U22583
ranimycin 10850 Rancomycin 2, U-25,873, U-25873
razupenem 10851 PZ-601, SM-216601, SMP-601
relebactam Approved drug 10852 MK-7655, MK-7655A, MK7655
retapamulin Approved drug 11035 Altabax®, Altargo®, SB-275833, SB275833
ribostamycin PDB Ligand 12161 SF-733
ridinilazole PDB Ligand 10853 SMT-19969, SMT19969
rifabutin Approved drug 12015 LM 427, Mycobutin®, Rifabutine
rifampicin Approved drug PDB Ligand 2765 Rifadin®, rifampin
rifamycin SV Approved drug 4570 Aemcolo®
rifapentine Approved drug PDB Ligand 12014 DL 473, MDL 473, Priftin®
rifaquizinone 11028 CBR-2092, TNP-2092
rifasutenizol 12959 TNP-2198
rifaximin Approved drug PDB Ligand 12012 L/105, Rifamycin L 105, Xifaxan®
ritipenem 10854 FCE-22101, FCE22101
Ro-406890 11048 ceftrazonal, Ro 40-6890, Ro 406890, Ro406890
rokitamycin Approved drug 12879 Ricamycin®, TMS-19-Q
rolitetracycline Approved drug 12760 pyrrolidinylmethyltetracycline, Reverin®, SQ 15,659, Syntetrin®, Velacycline®
rosaramicin 10855 Antibiotic 67-694, Antibiotic 67694, rosamicin, SCH-14947, SCH14947
rosoxacin Approved drug 12474 acrosoxacin, Eracine®, Eradacil®, Eradacin®, WIN 35213, Winuron®
roxithromycin Approved drug PDB Ligand 1465 RU 28965
RP60556A 11006
RS-102895 PDB Ligand Immunopharmacology Ligand 779 abaucin, RS102895
rufloxacin Approved drug 12473 MF 934, Monos®
 
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sanfetrinem 10856 GV104326
sarafloxacin Approved drug 10857 A-56620, A56620
sarecycline Approved drug PDB Ligand 12921 P005672, Seysara®
Sch 29482 11031
SCH-79797 10971 SCH 79797, SCH79797
secnidazole Approved drug 12925 14,539 RP, Solosec®, SYM-1219
SEQ-9 PDB Ligand 13159
sisomicin Approved drug PDB Ligand 10858 Antibiotic 66-40, Antibiotic 6640, rickamicin, Sch-13475, Sch13475, sisomycin, Sissomicin
sitafloxacin Approved drug 11040 compound 33 [PMID: 7932562], DU-6859, DU-6859a, DU6859a, Gracevit®, STX
SK&F 88070 11049 Skf 88070
solithromycin PDB Ligand 10859 CEM-101, CEM101, compound 3 [PMID: 30258539], OP-1068, OP1068, Solithera, T-4288, T4288
sorangicin A PDB Ligand 11038 (+)-Sorangicin A
sparfloxacin Approved drug 10860 AT-4140, AT4140, CI-978, CI978, SPFX, Zagam ®
spectinomycin Approved drug PDB Ligand 11127 actinospectacin, M-141, Trobicin®, U-18409, U-18409E, U18409
spenolimycin 10961 acmimycin
SPR741 13250 NAB741
SQ-109 Antimalarial Ligand 7997 MMV687273, SQ 109, SQ109
squalamine 10861 7alpha-Hydroxy, 3beta-spermidine, MSI-1256F (squalamine lactate)
SRI-20864 10986 SRI20864
SRI-20920 10987 SRI 20920, SRI20920
streptomycin Approved drug PDB Ligand 10923 Gerox®, NSC-14083, Strepcen®
SU-3327 10703 compound 9 [PMID: 19271755], halicin, SU3327
sudapyridine 13002 WX-081
sulbactam Approved drug PDB Ligand 10769 Betamaze, CP-45,899, CP-45899
sulbenicillin 12273 SBPC
sulfabenzamide Approved drug PDB Ligand 12632
sulfacetamide Approved drug 12633 Bleph-10®, Klaron®, sulphacetamide
sulfachlorpyridazine Approved drug 12634 BA-10370, sulfachloropyridazine, sulphachlorpyridazine
sulfadiazine Approved drug 12635
sulfadimethoxine Approved drug 12638 Albon® (veterinary), sulfadimethoxydiazine, sulphadimethoxine
sulfadimidine Approved drug 12642 sulfamethazine
sulfadoxine Approved drug Antimalarial Ligand 10173 sulphadoxine
sulfaguanidine Approved drug PDB Ligand 12639 sulfanilylguanidine, sulphaguanidine
sulfalene Antimalarial Ligand 10174 Kelfizine®, sulfamethopyrazine, sulfamethoxypyrazine, sulfametopyrazine
sulfamerazine Approved drug 12640 2-sulfanilamido-4-methylpyrimidine, sulfamethyldiazine, sulphamerazine
sulfamethizole Approved drug 12683 Rufol®, sulphamethizole, Thiosulfil®
sulfamethoxazole Approved drug PDB Ligand 10933 Gantanol®, RO 4-2130, RO-42130, SMX, STX-608
sulfamethoxypyridazine Approved drug 12686 Kynex®, sulphamethoxypyridazine
sulfametomidine 12701 methofadin, sulfamethomidine
sulfametoxydiazine Approved drug 12641 sulfameter, sulfamethoxydiazine, Sulla®
sulfametrole Approved drug 12702
sulfamonomethoxine Approved drug PDB Ligand 12688 Daimeton®
sulfamoxole Approved drug 12744 Nuprin®, sulfadimethyloxazole, Sulfuno®, sulphamoxole
sulfanilamide Approved drug PDB Ligand 12631 AVC®, sulphanilamide
sulfaperin 12742 Sulfaperine
sulfaphenazole 11352 Sulfabid®
sulfapyridine Approved drug PDB Ligand 12698 Dagenan®, M&B 693, sulphapyridine
sulfasalazine Approved drug PDB Ligand 4840 Azulfidine®, Salazopyridin®, Salazopyrin®, SAS-500
sulfathiazole Approved drug PDB Ligand 12699 M&B 760, Thiazamide®
sulfathiourea 12745 sulfathiocarbamide
sulfisoxazole Approved drug 12700 Gantrisin®, NU-445, sulfafurazole, sulphafurazole
sulopenem 10862 CP-70,429, CP-70429, CP70429
sultamicillin Approved drug 12290 CP-49,952, Unasyn®
sutezolid PDB Ligand 12772 MMV688756, PF-02341272, PNU-100480, U-100480
 
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tacapenem 10863 R-95867, R95867
talampicillin Approved drug 12289 BRL 8988, Talpen®
taniborbactam PDB Ligand 10774 VNRX-5133, VNRX5133
taurolidine Approved drug 13030 Defencath® (taurolidine + heparin), taurolin
tazobactam 10789 CXA-201, CXA201, YTR 830, YTR 830H, Zerbaxa® (ceftolozane + tazobactam)
TBA-7371 13133 AZ-7371, compound 1 [PMID:24957839], TBA7371
TBAJ-587 13060 compound 8 [PMID: 30803745]
TBAJ-876 PDB Ligand 13132 compound 46 [PMID: 30803745]
TBI-166 12961 pyrifazimine
TBI-223 13029
tebipenem pivoxil Approved drug 10864 L-084, LJC 11,084, LJC-11,084, LJC-11084, Orapenem®, TBPM-PI
tedizolid Approved drug PDB Ligand 10865 DA-7157, previously torezolid, Sivextro®, TR-700, TR700
teicoplanin Approved drug 10924 Antibiotic 8327A, MDL-507, Targocid®, teichomycin, teicoplanin A2
teixobactin 10972 compound of formula II [WO2014089053A1], N-[N-Methyl-D-Phe-Ile-Ser-D-Gln-D-aIle-Ile-Ser-]cyclo[D-Thr*-Ala-[3-(2-iminoimidazolidine-4beta-yl)-Ala-]-Ile-]
telacebec PDB Ligand 12953 MMV687696, Q203
telavancin Approved drug 10925 TD-6424, TD6424, Vibativ®
telithromycin Approved drug 10878 HMR-3647, Ketek®, Levviax®, RU-66647, RU66647
temafloxacin Approved drug 10866 A-62254, A62254, Abbott 62254, Omniflox®
temocillin Approved drug 10926 BRL-17421, BRL17421, Negaban®
tetracycline Approved drug 10927 achromycin, Ala-Tet®, Brodspec®, NSC-108579, Panmycin®, Sumycin®, TCN
tetroxoprim 12328
tevenel 12398
thiamphenicol PDB Ligand 12400
Thiazomycin A 10990 compound 6 [PMID: 18804380]
thioridazine Approved drug 100 Mellaril®, thioridazin, TP-21
ticarcillin Approved drug 10928 BRL-2288, BRL2288, Ticar, Timentin® (ticarcillin + clavulanate)
tigecycline 10929 GAR-936, GAR936, Tygacil®, WAY-GAR-936
tigemonam 10867 SQ-30213, SQ-30836 (tigemonam dicholate), SQ30213, SQ30836 (tigemonam dicholate)
timcodar 10868 VX-853, VX853
tinidazole Approved drug 12341 CP 12574, Fasigyn®, Tindamax®
tirandalydigin 11012
tobramycin Approved drug PDB Ligand 10930 Bethkis®, Kitabis®, Tobi Podhaler®, Tobradex® (tobramycin + dexamethasone), Vantobra®
tomopenem 10869 CS-023, CS023, R-115685, R115685, RO-4908463
tosufloxacin Approved drug 12878 Ozex®, T-3262
TP-271 11013 TP271
TP-6076 PDB Ligand 13198
trimethoprim Approved drug PDB Ligand 10931 BW-56-72, BW-5672, NSC-106568, Primsol®, Proloprim®, Trimpex®
troleandomycin Approved drug 10209 oleandocetin, Tao®, triacetyloleandomycin
trospectomycin 10870 U-63,366F, U-63366F, U63366F
TXA6101 PDB Ligand 13012
TXA709 13160
 
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upleganan 12797 compound 44 [PMID: 31525992], EVER206, SPR206
 
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vaborbactam Approved drug PDB Ligand 10871 compound 9f [PMID: 25782055], RPX-7009, RPX7009, Vabomere (vaborbactam + meropenem)
vancomycin Approved drug 10932 Vancocin®, Vancor®
vanillobiocin 12130 novclobiocin 311
verapamil Approved drug 2406 Ansyr®, CP-165331 / CP-16533-1, Securon®
verdamicin 11010 6'-C-Methylsisomicin
vermisporin 11011
vertilmicin 11018
viomycin Approved drug 13252 celiomycin, florimycin, tuberactinomycin B
viquidacin 10872 AVE-4221, AVE4221, compound 1 [PMID: 23968485], NXL-101, NXL101
 
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walrycin B 11256
 
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xeruborbactam PDB Ligand 13131 QPX7728
 
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zabofloxacin 10873 DW-224a
zidebactam 10874 WCK-5107, WCK5107
zifanocycline 12794 KBP-7072
zoliflodacin PDB Ligand 10875 AZD-0914, AZD0914, EXT-0914, EXT0914
zosurabalpin PDB Ligand 12950 Abx MCP, RG6006, RO7223280