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The IUPHAR/BPS Guide to PHARMACOLOGY complete ligand list

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Ligand name ID Synonyms
A Back to top
A2315A 10846
acorafloxacin 10753 avarofloxacin (former name), JNJ-Q2, JNJQ2
ACX-362E 11030 ACX362E, ibezapolstat
afabicin 10754 Debio 1450, Debio1450
alalevonadifloxacin 10756 WCK 2349, WCK-2349, WCK2349
Altromycin B 10964
amifloxacin 10758 compound 7 [PMID: 2834557], WIN 49, 375, WIN 49,375-3, WIN-49375, WIN49375
amikacin Approved drug PDB Ligand 10894 Amikin®, AMK, Arikayce liposomal®, BB-K8
amoxicillin Approved drug 10895 Amoxil®, BRL-2333, co-amoxiclav (amoxicillin + clavulanic acid), Moxatag®, NSC-277174, Trimox®
ampicillin Approved drug PDB Ligand 10896 aminobenzylpenicillin, KS-R1, Penbritin®, Polycillin, Principen®
AN0128 10983 AN 0128, AN-0128, compound 2g [PMID: 16997550]
apalcillin 10759 PC-904, PC904, WY-44,417, WY-44417
apramycin PDB Ligand 10760 EL-857, EL857, Nebramycin factor 2, Nebramycin II
arbekacin PDB Ligand 7345 arbekacin sulfate, ME1100, NPC-14
avibactam Approved drug PDB Ligand 10761 AVI, NXL 104, NXL-104, NXL104
azithromycin Approved drug PDB Ligand Antimalarial Ligand 6510
aztreonam Approved drug 10763 Azactam®, Cayston®, SQ 26776, SQ-26776, SQ26776
 
B Back to top
BAL19403 10981 BAL 19403, BAL-19403
BAL30072 11004 BAL-30072
BAS-118 10976 BAS118, compound 7n [PMID: 11728192]
BC-3205 10998
BC-7013 11034 BC7013
bederocin PDB Ligand 10764 REP-8839, REP8839
BLI-489 free acid 10995 BLI489
bluensomycin 10765 bluensin, U-12898, U12898
borrelidin Antimalarial Ligand 11306 (-)-borrelidin
BRL-42715 10993 C6-(N1-Methyl-1,2,3-trazolylmethylene)penem, LS-186900 (sodium salt), LS-187554
BRL-44154 11036 analogue 4f [Brown et al., 1991], BRL44154
butikacin 10766 UK-18,892, UK-18892, UK18892
 
C Back to top
cadazolid PDB Ligand 10767 ACT-179811, ACT179811
caffeic acid PDB Ligand 5155
carbenicillin Approved drug 10768 BRL-2064, BRL2064, carboxybenzylpenicillin, CBPC, CP 15639-2, CP-156392, Pyopen®
cationomycin 11002 BRN-6263205, BRN6263205, LS-52659, LS52659
CB-182804 11003 CB-182,804, CB182804
cefaclor Approved drug 10897 Ceclor®, Lilly 99638, Raniclor®
cefadroxil Approved drug 4831 Duricef®
cefazaflur 10770 SK&F 59962
cefazolin 10935 Ancef®, cephazolin, CEZ, Kefzol®, SK&F-41558
cefclidin 10771 cefclidine, E-1040, E1040
cefepime Approved drug 10772 BMY-28142, BMY28142, CFPM, Maxipime®, Renapime®
cefetecol 10775 GR-69153, GR-69153X, GR69153
cefiderocol Approved drug 10776 compound 3 [PMID: 29960205], Fetcroja®, Fetroja®, GSK-2696266, GSK2696266, RSC 649266, RSC-649266, RSC649266, S-649266
cefixime Approved drug PDB Ligand 10898 (E)-Cefixime, Cefspan®, CFIX, FK-027, FR-17027, Suprax®
cefluprenam 10777 E-1077, E1077
cefmatilen 10778 S-1090, S1090
cefotaxime Approved drug PDB Ligand 10893 Claforan®, Ru-24756
cefotetan Approved drug 10936 Apatef®, Cefotan®, ICI-156834, ICI156834
cefoxitin Approved drug PDB Ligand 10937 Cenomycin®, CFX, Mefoxin®, MK-306, MK306
cefpimizole 10779 CPIZ, U 63196E, U-63,196, U-63196E
cefpodoxime Approved drug 10780 RU-51746, Vantin®
cefsulodin 10783 Cefonomil®, CGP-7174-E, CGP7174/E
ceftaroline fosamil Approved drug 10899 PPI-0903, TAK-599, Teflaro®, Zinforo®
ceftazidime Approved drug 10762 CAZ, Fortaz®, Fortum®, GR 20263, GR-20263, GR20263, LY-139381, LY139381, Pentacef®, Tazicef®
cefteram 11051 cefetamet, cefteram pivoxil (prodrug), CFTM, Ro 19-5247, T-2525
ceftiolene 10784 42980RP, cefatiolene, RP 42,980, RP 42980, RP-42980, RP42980
ceftizoxime Approved drug 10785 Cefizox®, compound 22 {PMID: 2342058], Epocelin®, FK-749, FK749, FR-13749, FR13749, SK&F 88373-Z
ceftizoxime alapivoxil 10786 AS-924, AS924, KY-020, KY020
ceftobiprole Approved drug 10787 BAL-9141, BAL9141, BAL9141-000, BAL9141000, Ro-63-9141, Ro-639141, Zeftera®, Zevtera®
ceftolozane Approved drug 10788 CXA-101, CXA101, FR-264205, FR264205, Zerbaxa® (ceftolozane + tazobactam)
ceftriaxone Approved drug 5326 Rocephin®
cefuroxime Approved drug PDB Ligand 10900 Ceftin®, CXM, Kefurox®, Zinacef®
cephalexin Approved drug 4832 cefalexin, Ceporex®, Keflex®
cephradine Approved drug 4830 cefradine, Infexin®, Velocef®
cetefloxacin 10790 compound 43f [PMID: 7990118], E-4868, E4868
cethromycin PDB Ligand 10791 A-195773, Abbott-195773, ABT-773, ABT773, Restanza®
cetocycline 10792 A-40728, Abbott 40728, chelocardin, compound 1 [PMID: 379332]
CG-400549 PDB Ligand 10984 CG400549
CGP-31608 10963 CGP 31608, CGP31608
chalcomycin 11058
chinfloxacin 11017
chloramphenicol Approved drug PDB Ligand 10901 Brolene®
chlorocardicin 11044
chrysin PDB Ligand 8789 NSC-407436
cilastatin Approved drug 5166 MK 0791, MK-791, MK791, Primaxin®
ciprofloxacin Approved drug PDB Ligand 10902 BAY-O-9867, BAY-O9867, Cetraxal®, Ciloxan®, Cipro®, CPFX, Proquin XR
CJ-15,801 Antimalarial Ligand 10610 CJ-15801
cladosporin PDB Ligand Antimalarial Ligand 10247 asperentin
clarithromycin Approved drug PDB Ligand 10903 6-O-methylerythromycin, A-56268, ABBOTT-56268, Biaxin®, Klaricid®, TE-031
clinafloxacin 10793 AM 1091, CI-960, PD-127321
clindamycin Approved drug PDB Ligand Antimalarial Ligand 10607
colistin Approved drug 10794 Colobreathe®, polymyxin E, Promixin®
compound 2 [PMID: 33085774] Antimalarial Ligand 11322
contezolid PDB Ligand 10795 MRX-1, MRX-I
contezolid acefosamil (parent) 10796 MRX-4
Corallopyronin A 11029 CorA, LS-54950, LS54950
coumamycin PDB Ligand 10879 coumermycin A1, notomycin
CRS3123 PDB Ligand 10991 CRS-3123, REP-3123, REP3123
cyclothialidine 10988 Ro 09-1437
 
D Back to top
dactimicin 11001 Formimidoyl-fortimicin A, SF-2052, SF2052
dalbavancin Approved drug 10876 BI-397, BI397, Dalvance®, Xydalba®
dalfopristin Approved drug PDB Ligand 10797 RP-54476, RP54476, Synercid® (dalfopristin + quinupristin)
danirixin Immunopharmacology Ligand 8500 GSK-1325756B, GSK1325756, GSK1325756B
dapsone Approved drug Antimalarial Ligand 10934 Aczone®, NSC-6091
daptomycin Approved drug 10904 Cubicin®, LY-146032, LY146032
DC-159a 10982
DEBIO 1452 10755 afabicin desphosphono, AFN-1252, AFN-12520000, DEBIO-1452, DEBIO1452
decaplanin 10968 M 861410, M86-1410, MM-47761
delafloxacin Approved drug 10799 Abbott 492, ABT-492, ABT492, Baxdela®, Quofenix®
delpazolid 10999 LCB-01,0371, LCB-01-0371, LCB01-0371
demeclocycline 10905 Declomycin®, Ledermycin®
diacerein Approved drug 10800 Artrodar®, Fisiodar®
difficidin 11062
difloxacin 10801 A 56619, A-56619, Dicural®
dihydroxybenzofuran 10992 2,3-Benzofurandiol
DK-507k 11037
doxycycline Approved drug PDB Ligand Immunopharmacology Ligand Antimalarial Ligand 6464 BMY-28689, Monodox®, Vibramycin®
DS-8587 10955 DS8587
DS-2969b 10985 DS 11960558 (DS-2969b prodrug), DS-2969, example 2 [WO2017/056012A1]
Dup-105 10950 DuP 105, DuP105
DuP-721 10960 DuP 721
DX-619 11039 compound 4 [PMID: 19736016], DX619
 
E Back to top
E-0702 11056
ecenofloxacin 10802 CFC-222, CFC222
E-1010 free base 11050 E1010, ER-35786
Enduracidin 10989
enoxacin Approved drug 8882 AT-2266, CI-919, Penetrex®
enteromycin carboxamide 11063 BRN 2416858, BRN-2416858, BRN2416858, LS-14645
eperezolid 10803 comound 2 [PMID: 23584544], PNU-100592, PNU100592, U-100592, U100592
epicillin 10804 Dexacillin®, SQ 11302, SQ-11302, SQ11302
eravacycline Approved drug PDB Ligand 10805 compound 17j [PMID: 2148514], TP-434, TP434, Xerava®
eremomycin 10959 A82846A
ertapenem Approved drug 10906 Invanz®, L-749345, MK-0826, MK-826
erythromycin Approved drug PDB Ligand 1456 EM-A, E-Mycin®, Erythrocin®, erythromycin-A
etheromycin 10994 CP‐38 295
ethyl bromopyruvate 10952
ETX0282 10781 ETX-0282
ETX1317 10782 ETX-1317
evernimicin 10806 SCH 27899, SCH-27899, SCH27899, Ziracin®
 
F Back to top
fandofloxacin 10807 DW-116, DW116
faropenem PDB Ligand 10808 compound 1 [PMID: 9216830], faropenem medoxomil, fropenem
feldamycin 10979 BMY-28565, BMY28565, U-48266
Ferrimycin A1 10966
ficellomycin 10965 U-47,929, U-47929, U47929
fidaxomicin Approved drug PDB Ligand 10909 Dificid®, Dificlir®, OPT-80, PAR-101
finafloxacin 10809 AL-60371, AL60371, Xtoro®
flucloxacillin Approved drug 10910 BRL-2039, BRL2039, floxacillin
fludalanine 10810 3-fluoro-D-alanine, MK-0642, MK0642
fosfomycin Approved drug PDB Ligand 10813 Monurol®, phosphomycin, phosphonomycin, Veramina®
fosmidomycin PDB Ligand Antimalarial Ligand 9739 FR-31564
furazolium 10814 Novofur
fusidic acid Approved drug PDB Ligand 10815 CEM-102, CEM102, Fucidin®, fusidate, sodium fusidate, Taksta®
 
G Back to top
gatifloxacin Approved drug 10816 AM-1155, AM1155, Gatiflo®, GTFX, Tequin®, Zymar®
gentamicin Approved drug 2427 Garamycin®, gentamicin sulfate
gepotidacin PDB Ligand 10817 GSK-2140944, GSK2140944
gloximonam 10880 SQ 82,291, SQ 82531, SQ-82531, SQ82531
grepafloxacin Approved drug 10818 OPC 17116, OPC-17116, OPC17116, Raxar®
 
H Back to top
hedamycin 10958 antibiotic B 26,158, B26158, NSC-70929
hesperetin PDB Ligand 10953 3',5,7-Trihydroxy-4'-methoxyflavanone, NP-13, NSC-57654
hexachlorophene Approved drug PDB Ligand 11069 Inh 1 [PMID: 32284327], Nabac®
ω-Hydroxyemodin 11005 Citreorosein, omega-Hydroxyemodin
 
I Back to top
ibafloxacin 10819 R-835, R835, S-25930, S25930
iclaprim 10820 AR-100, AR100, Mersarex®, RO-48-2622, RO-482622
imipenem Approved drug 10821 MK-0787, MK0787, Primaxin® (imipenem + cilastatin), Recarbrio® (imipenem + cilastatin + relebactam).
indanomycin 10949 X-14547A
indolmycin PDB Ligand Antimalarial Ligand 11021 PA 155 A, PA-155-A, PA-155A, TAK-083
Irresistin-16 10973 IRS-16, IRS16
iseganan 10822 IB-367, IB-367-03
IT-62-B 11032
ivermectin Approved drug 2373 Heartgard®, ivermectin B1a, MK-933, Sklice®, Soolantra®
 
K Back to top
kaempferol PDB Ligand 11052 Robigenin
Katanosin B 10970 Lysobactin
KB-5246 11046 KB5246, LS-99630
kibdelomycin A 11016
 
L Back to top
L-701677 11042 L-701,677
L-708365 10980 L 708,365, L 708365, L-708,365
lactivicin 11022 compound 1 [PMID: 17676039], LTV
lascufloxacin 10823 KRP-AM1977
LBM-415 11043 LBM415, NVP LBM-415, NVP-PDF-713, PDF-713
lefamulin Approved drug PDB Ligand 10824 BC-3781, BC3781, compound 7 [PMID: 24874438], Xenleta®
leinamycin 11041 DC-107, DC107
lenapenem 10825 BO-2727, BO2727, L-739,428, L-739428
levofloxacin Approved drug PDB Ligand 10911 DR-3355, Levaquin®, Quinsair®
levonadifloxacin 10757 (S)-(-)-nadifloxacin, WCK 771, WCK-771, WCK771
levopropicillin 10826 BRL-284, BRL284, L-Propicillin, P-248, P248
lincomycin Approved drug PDB Ligand 10941 Bactramycin®, L-Mycin®, LCM, Lincocin®, Lincorex®, U 10,149A, U-10149
linezolid Approved drug PDB Ligand 10827 PNU-100766, PNU100766, U-100,766, U-100766, ZLD, Zyvox®
luminamicin 11053 coloradocin, LS-90907
lymecycline Approved drug 10912 N-Lysinomethyltetracycline, tetracycline-L Methylene-Lysine, Tetralysal®
lysinomicin 10969
 
M Back to top
M14659 11047 GR 63116, GR-63116, M 14659, M-14659
Macquarimicin A 10978
maridomycin 10828 LS-87912, Maridomycin III
MC-02479 11033 MC 02479, MC02479, RWJ 54428, RWJ-54428
ME-1228 acid 11045 ME1228
meropenem PDB Ligand 10829 ICI 194,660, Merrem®, SM-7338
mersacidin 11014 M87 1551, M87-1551
methenamine Approved drug 10913 Hiprex®, Mandelamine®, Urex®
metronidazole Approved drug PDB Ligand 10914 BAY-5360, BAYER 5360, Flagyl®, Metrogel®, ROZEX®
MGB-BP-3 10996 compound 50 [PMID: 17960927], MGB-BP3
mideplanin 10830 CTA A1, MDL 62873, MDL-62873, MDL62873
minocycline Approved drug 10831 CL 59806, CL-59806, CL59806, Dynacin®, MINO, Minocin®, NSC-141993
moxifloxacin Approved drug PDB Ligand 10915 Avelox®, BAY-12-8039, BAY-128039, BAY128039, MFX, MOXIVIG® (opthalmic solution)
mupirocin Approved drug Antimalarial Ligand 10916 Bactroban®, BRL-4910A, BRL-4910F, Centany®
murepavadin 10832 POL7080, RG-7929, RG7929, RO-7033877, RO7033877
MUT056399 PDB Ligand 11000 Fab-001, FAB001, MUT-056399
 
N Back to top
nacubactam 10833 OP-0595, OP0595, RG-6080, RG6080, RO-7079901, RO7079901
nafcillin Approved drug 10942 Ethoxynaphthamido Penicillin Sodium, Nallpen®, Unipen®
nafithromycin 10834 WCK 4873, WCK-4873, WCK4873
napsamycin C 11008
napsamycin D 11009
narasin 10835 C-7819B, Lilly 79891, Monteban®, Narasin A
nemonoxacin Approved drug 10836 Taigexyn®, TG-873870, TG873870
neomycin Approved drug PDB Ligand 709 Neo-Rx®, neomycin sulfate
neopyrrolomycin 10962
nifurprazine 10837 carofur, HB-115, HB115
nitrofurantoin Approved drug PDB Ligand 10917 Furadantin®, Macrobid®, Macrodantin®, Nitro Macro®, NSC-2107, NSC-44150
nodusmicin 11019 nodusmicin 1
nojirimycin 10951 5-amino-5-deoxy-D-glucopyranose, D-gluco-piperidinose
NSC-84963 10956 NSC 84963, NSC84963
NSC-93169 10957 NSC 93169, NSC93169
 
O Back to top
ofloxacin Approved drug 10918 DL-8280, Exocin® (eye drops), Floxin®, HOE-280, OFX, Tarivid®
olamufloxacin 10838 HSR-903, HSR903
oleuropein 11027
omadacycline Approved drug 10839 amadacycline, compound 6 [PMID: 21302930], Nuzyra®, PTK-0796, PTK0796
oritavancin Approved drug 10877 Kimyrsa®, LY-333328, LY333328, Orbactiv®
oxacillin Approved drug 10943 Bactocill®
oxantel Approved drug 10840 CP-14,445, CP-14445
oxaquin 10997 DNV-3837, DNV3837, MCB-3837, MCB3837
oxytetracycline Approved drug PDB Ligand 10919 E703, NSC-9169, Terramycin®
ozenoxacin Approved drug 10841 Ozadub®, T-3912, T3912, Xepi®
 
P Back to top
pafuramidine 10842 DB-289, DB289
paldimycin 10843 Antibiotic 273 A, U-70,138, U-70138F
penicillin G Approved drug PDB Ligand 4796 penicillin G sodium, penicillin-G potassium
phenoxymethylpenicillin Approved drug PDB Ligand 10920 Oracillin®, PC Pen VK®, Pen-V®, penicillin V, Penicillin VK, PNV
phleomycin 10954 NSC 61586, NSC-61586
piperacillin Approved drug PDB Ligand 10921 CL 227,193, CL-227193, PIPC, T-1220, Tazocin® (piperacillin + tazobactam)
pirazmonam 10844 compound 2 [PMID: 25658376], SQ 83,360, SQ-83360, SQ83360
pirbenicillin 10845 CP-33,994, CP-33,994-2
pivmecillinam Approved drug 10922 amdinocillin pivoxil, pivmecillinam hydrochloride, RO-10-9071, RO-109071, Selexid®
plazomicin Approved drug PDB Ligand 10847 ACHN-490, ACHN490, Zemdri®
plusbacin A3 11020
PNU-288034 10977 compound 2 [PMID: 16644216], PNU288034
poststatin 10967 L-Val-L-Val-3-amino-2-oxo-valeryl-D-Leu-L-Val
premafloxacin 10848 compound 21 [PMID: 17303420], U-95376, U95376
 
Q Back to top
quinupristin Approved drug 10798 RP 57669, RP-57669, RP57669, Synercid® (dalfopristin + quinupristin)
 
R Back to top
radezolid PDB Ligand 10849 Rx-01_667, RX-103, RX-1741, RX103, RX1741
ranbezolid 11007 RBx 7644
rancinamycin IA 11015 Rancomycin 1, U-22583, U22583
ranimycin 10850 Rancomycin 2, U-25,873, U-25873
razupenem 10851 PZ-601, SM-216601, SMP-601
relebactam Approved drug 10852 MK-7655, MK-7655A, MK7655
retapamulin Approved drug 11035 Altabax®, Altargo®, SB-275833, SB275833
ridinilazole 10853 SMT-19969, SMT19969
rifampicin Approved drug PDB Ligand 2765 Rifadin®, rifampin
ritipenem 10854 FCE-22101, FCE22101
Ro-406890 11048 ceftrazonal, Ro 40-6890, Ro 406890, Ro406890
rosaramicin 10855 Antibiotic 67-694, Antibiotic 67694, rosamicin, SCH-14947, SCH14947
RP60556A 11006
 
S Back to top
sanfetrinem 10856 GV-118819, GV-118819X, GV118819
sarafloxacin Approved drug 10857 A-56620, A56620
Sch 29482 11031
SCH-79797 10971 SCH 79797, SCH79797
sisomicin PDB Ligand 10858 Antibiotic 66-40, Antibiotic 6640, Sch-13475, Sch13475, sisomycin, Sissomicin
sitafloxacin Approved drug 11040 compound 33 [PMID: 7932562], DU-6859, DU-6859a, DU6859a, Gracevit®, STX
SK&F 88070 11049 Skf 88070
solithromycin PDB Ligand 10859 CEM-101, CEM101, compound 3 [PMID: 30258539], OP-1068, OP1068, Solithera, T-4288, T4288
sorangicin A PDB Ligand 11038 (+)-Sorangicin A
sparfloxacin Approved drug 10860 AT-4140, AT4140, CI-978, CI978, SPFX, Zagam ®
spenolimycin 10961 acmimycin
SQ-109 Antimalarial Ligand 7997 MMV687273, SQ 109, SQ109
squalamine 10861 7alpha-Hydroxy, 3beta-spermidine, MSI-1256F (squalamine lactate)
SRI-20864 10986 SRI20864
SRI-20920 10987 SRI 20920, SRI20920
streptomycin